SCHEMBL8889934

SCHEMBL8889934

COc1cc(CS(=O)(=O)C(C)C)ccc1CNc1nc(Nc2ccc(Cl)cc2)c2cc(C)ccc2n1

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CTNNB1 P35222 13/20 0.46
TCF7L2 Q9NQB0 13/20 0.46
P2RX3 P56373 1/20 0.43
GRK6 P43250 2/20 0.42
SLC2A1 P11166 1/20 0.41
NTRK1 P04629 2/20 0.38
PDE5A O76074 1/20 0.38
AURKA O14965 1/20 0.38
IGF1R P08069 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8889431 0.72 EGFR (0.43) CTNNB1TCF7L2P2RX3
SCHEMBL8891133 0.72 NPY5R (0.46) CTNNB1TCF7L2PDE5A
SCHEMBL4170114 0.63 CTNNB1 (1.00) CTNNB1TCF7L2
SCHEMBL4174294 0.61 CTNNB1 (0.78) CTNNB1TCF7L2
SCHEMBL30380040 0.60 CYP1A2 (0.56)
SCHEMBL20682390 0.60 L3MBTL1 (0.46)
SCHEMBL4160385 0.59 CTNNB1 (1.00) CTNNB1TCF7L2
SCHEMBL6039137 0.59 NPY5R (0.57) SLC2A1
SCHEMBL5569927 0.59 KDM4E (0.74)
SCHEMBL7254867 0.59 PIN1 (0.57) PDE5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997020822-A1 QUINAZOLIN-2,4-DIAZIRINES AS NPY RECEPTOR ANTAGONIST NOVARTIS AG (CH) 1997-06-12 WO disclosed