SCHEMBL8889431

SCHEMBL8889431

COCc1cc(CS(=O)(=O)C(C)C)ccc1Nc1nc(Nc2ccc(Cl)cc2)c2cc(N(C)C)ccc2n1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
EGFR P00533 3/20 0.43
NPY5R Q15761 5/20 0.39
KDR P35968 2/20 0.36
CTNNB1 P35222 5/20 0.34
TCF7L2 Q9NQB0 5/20 0.34
P2RX3 P56373 3/20 0.34
KDM1A O60341 2/20 0.33
PIN1 Q13526 1/20 0.33
ALDH1A1 P00352 1/20 0.33
GAA P10253 1/20 0.33
MAPT P10636 1/20 0.33
MAPK1 P28482 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8891648 0.76 NPY5R (0.41) EGFRNPY5RCTNNB1TCF7L2
SCHEMBL8889934 0.72 CTNNB1 (0.46) CTNNB1TCF7L2P2RX3
Hydrochloric Acid SCHEMBL8889724 0.68 NPY5R (0.76) EGFRNPY5RKDM1AL3MBTL1
SCHEMBL8891133 0.67 NPY5R (0.46) NPY5RKDRCTNNB1TCF7L2MAPT
SCHEMBL8893267 0.65 NPY5R (0.60) EGFRNPY5RKDM1AALDH1A1L3MBTL1
SCHEMBL8890735 0.64 EGFR (0.63) EGFRNPY5RKDM1AMAPTMAPK1
Hydrochloric Acid SCHEMBL8909035 0.64 NPY5R (0.59) EGFRNPY5RKDM1AALDH1A1L3MBTL1
Hydrochloric Acid SCHEMBL8888779 0.64 EGFR (0.62) EGFRNPY5RKDM1AMAPTMAPK1
SCHEMBL7254867 0.59 PIN1 (0.57) EGFRNPY5RKDRPIN1MAPT
SCHEMBL8891909 0.58 NPY5R (0.83) EGFRNPY5R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997020822-A1 QUINAZOLIN-2,4-DIAZIRINES AS NPY RECEPTOR ANTAGONIST NOVARTIS AG (CH) 1997-06-12 WO disclosed