SCHEMBL8890558

SCHEMBL8890558

O=c1[nH]c2c(N3CCNCC3)cccc2n1C1CCCCC1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 1/20 0.55
CHRM1 P11229 2/20 0.49
CHRM2 P08172 1/20 0.49
CHRM4 P08173 1/20 0.49
CHRM3 P20309 1/20 0.49
OPRM1 P35372 6/20 0.47
OPRK1 P41145 4/20 0.47
OPRD1 P41143 2/20 0.47
OGFRL1 Q5TC84 1/20 0.47
OPRL1 P41146 5/20 0.44
ALDH1A1 P00352 4/20 0.41
PKM P14618 1/20 0.41
CYP3A4 P08684 2/20 0.41
CYP2C9 P11712 2/20 0.41
CYP2C19 P33261 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
MAPK1 P28482 2/20 0.41
NR5A2 O00482 1/20 0.41
LMNA P02545 1/20 0.41
TP53 P04637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22605719 0.83 HTR6 (0.47) HTR6CHRM1CHRM2CHRM4CHRM3
SCHEMBL8902683 0.80 CHRM2 (0.42) CHRM1CHRM2CHRM4CHRM3OPRM1
SCHEMBL31152738 0.78 HTR6 (0.50) HTR6CHRM2OPRM1ALDH1A1
SCHEMBL28512511 0.73 OPRM1 (0.43) CHRM1CHRM2CHRM4CHRM3OPRM1
SCHEMBL28514062 0.72 OPRM1 (0.39) HTR6CHRM1CHRM2CHRM4CHRM3
SCHEMBL22869704 0.72 HSD11B1 (0.52) ALDH1A1CYP3A4CYP2C19SMN1; SMN2MAPK1
SCHEMBL28497378 0.72 CHRM1 (0.42) HTR6CHRM1CHRM2CHRM4OPRM1
SCHEMBL4306275 0.72 CHRM1 (0.57) CHRM1OPRM1OPRL1DRD2KCNH2
SCHEMBL3243793 0.72 HSD11B1 (0.53) CHRM1CHRM2CHRM4CHRM3OPRM1
SCHEMBL3243652 0.72 OPRM1 (0.62) CHRM1OPRM1OPRK1OPRD1OPRL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997016187-A1 MUSCARINE ANTAGONISTS MERCK & CO., INC. (US) 1997-05-09 WO disclosed