SCHEMBL8891569

SCHEMBL8891569

COc1ccc(CCOc2cc(C(=O)O)ncc2OC)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.52
ASPH Q12797 1/20 0.52
RIOX2 Q8IUF8 1/20 0.52
KDM8 Q8N371 1/20 0.52
SIGMAR1 Q99720 1/20 0.45
CYP11B1 P15538 1/20 0.45
CYP11B2 P19099 1/20 0.45
CSNK2A2 P19784 1/20 0.44
CSNK2A1 P68400 1/20 0.44
CYP1A2 P05177 2/20 0.43
CYP3A4 P08684 2/20 0.43
CYP2C9 P11712 2/20 0.43
ALDH1A1 P00352 1/20 0.43
POLB P06746 1/20 0.43
HPGD P15428 1/20 0.43
CYP2C19 P33261 1/20 0.43
ATM Q13315 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
TRPC6 Q9Y210 2/20 0.43
PDGFRB P09619 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8888044 0.93 KDM4E (0.47) KDM4EASPHRIOX2KDM8SIGMAR1
SCHEMBL8893284 0.89 HTR2C (0.43) KDM4EASPHRIOX2KDM8SIGMAR1
SCHEMBL8890258 0.89 CYP1A2 (0.47) KDM4EASPHRIOX2KDM8SIGMAR1
SCHEMBL21045912 0.84 TRPC6 (0.57) KDM4EASPHRIOX2KDM8SIGMAR1
SCHEMBL10532890 0.83 KDM4E (0.55) KDM4EASPHRIOX2KDM8CYP1A2
SCHEMBL8890675 0.81 CYP11B1 (0.50) SIGMAR1CYP11B1CYP11B2CYP1A2CYP3A4
SCHEMBL8890275 0.80 PDE4D (0.57)
SCHEMBL21045700 0.78 TRPC6 (0.54) KDM4EASPHRIOX2KDM8TRPC6
SCHEMBL30439705 0.78 TRPC6 (0.54) KDM4EASPHRIOX2KDM8TRPC6
SCHEMBL8892821 0.78 KDM4E (0.47) KDM4EASPHKDM8CYP1A2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997003967-A1 SUBSTITUTED AROMATIC COMPOUNDS AND THEIR PHARMACEUTICAL USE RHONE-POULENC RORER LIMITED (GB) 1997-02-06 WO disclosed