SCHEMBL8891572

SCHEMBL8891572

c1ccc(COCCCOc2ccc(Nc3nc(Nc4ccccc4)c4ccccc4n3)cc2)cc1

nearest known ligand 0.60

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NPY5R Q15761 10/20 0.60
CHEK2 O96017 1/20 0.55
EGFR P00533 1/20 0.55
ERBB2 P04626 1/20 0.55
ROS1 P08922 1/20 0.55
FLT3 P36888 1/20 0.55
ERBB4 Q15303 1/20 0.55
AURKB Q96GD4 1/20 0.55
CLK4 Q9HAZ1 1/20 0.55
MKNK2 Q9HBH9 1/20 0.55
SLC2A1 P11166 1/20 0.54
PIN1 Q13526 1/20 0.51
MERTK Q12866 4/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8891002 0.91 NPY5R (0.54) NPY5RCHEK2EGFRERBB2ROS1
Hydrochloric Acid SCHEMBL8890646 0.91 NPY5R (0.53) NPY5RCHEK2EGFRERBB2ROS1
SCHEMBL8900235 0.91 NPY5R (0.61) NPY5REGFRERBB2AURKBCLK4
SCHEMBL8900305 0.88 EGFR (0.69) NPY5RCHEK2EGFRERBB2ROS1
SCHEMBL8891978 0.88 NPY5R (0.65) NPY5RSLC2A1PIN1MERTK
Hydrochloric Acid SCHEMBL8899588 0.87 CHEK2 (0.67) NPY5RCHEK2EGFRERBB2ROS1
SCHEMBL8891059 0.86 MERTK (0.66) NPY5RCHEK2EGFRERBB2ROS1
Hydrochloric Acid SCHEMBL8909111 0.85 MERTK (0.64) NPY5RCHEK2EGFRERBB2ROS1
SCHEMBL8891704 0.82 NPY5R (0.67) NPY5RSLC2A1PIN1MERTK
SCHEMBL8890861 0.82 NPY5R (0.77) NPY5RCHEK2EGFRERBB2ROS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997020822-A1 QUINAZOLIN-2,4-DIAZIRINES AS NPY RECEPTOR ANTAGONIST NOVARTIS AG (CH) 1997-06-12 WO claimed
WO-1997020822-A1 QUINAZOLIN-2,4-DIAZIRINES AS NPY RECEPTOR ANTAGONIST NOVARTIS AG (CH) 1997-06-12 WO disclosed