SCHEMBL8891975

SCHEMBL8891975

O=C(O)c1ccc2ccccc2c1Sc1ccccc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
WDR5 P61964 1/20 0.58
LDHA P00338 1/20 0.56
NR4A1 P22736 1/20 0.52
NR4A2 P43354 1/20 0.52
NR4A3 Q92570 1/20 0.52
MEN1 O00255 4/20 0.51
KMT2A Q03164 4/20 0.51
ALDH1A1 P00352 4/20 0.51
MAPT P10636 1/20 0.51
CDC25B P30305 1/20 0.46
HPGD P15428 4/20 0.44
PKM P14618 1/20 0.43
RAB9A P51151 1/20 0.43
RXFP1 Q9HBX9 1/20 0.43
LMNA P02545 1/20 0.43
CSNK2A2 P19784 1/20 0.43
CSNK2B P67870 1/20 0.43
CSNK2A1 P68400 1/20 0.43
KDM4E B2RXH2 2/20 0.42
GLA P06280 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6843928 0.91 WDR5 (0.63) WDR5LDHANR4A1NR4A2NR4A3
SCHEMBL599807 0.84 WDR5 (0.63) WDR5LDHANR4A1NR4A2NR4A3
SCHEMBL7542084 0.81 WDR5 (0.51) WDR5LDHANR4A1NR4A2NR4A3
SCHEMBL24723588 0.77 ALDH1A1 (0.56) NR4A1NR4A2NR4A3MEN1KMT2A
SCHEMBL23665075 0.74 ALDH1A1 (0.53) LDHAMEN1KMT2AALDH1A1MAPT
SCHEMBL895573 0.74 WDR5 (1.00) WDR5LDHANR4A1NR4A2NR4A3
SCHEMBL29721418 0.74 WDR5 (1.00) WDR5LDHANR4A1NR4A2NR4A3
SCHEMBL12427691 0.73 WDR5 (0.50) WDR5LDHANR4A1NR4A2NR4A3
Phenanthrene SCHEMBL29265471 0.73 NR4A1 (0.75) WDR5LDHANR4A1NR4A2NR4A3
Phenanthrene SCHEMBL31651179 0.73 NR4A1 (0.75) WDR5LDHANR4A1NR4A2NR4A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997048672-A2 SUBSTITUTED TETRAHYDRONAPHTHALENE AND DIHYDRONAPHTHALENE DERIVATIVES HAVING RETINOID AND/OR RETINOID ANTAGONIST-LIKE BIOLOGICAL ACTIVITY ALLERGAN SALES, INC. (US) 1997-12-24 WO disclosed