SCHEMBL8892237

SCHEMBL8892237

CC(C)(C)OC(=O)NC(Cc1ccccc1)C(CC(Cc1cccc(F)c1)C(=O)O)O[Si](C)(C)C(C)(C)C

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSS P25774 4/20 0.49
CTSK P43235 3/20 0.49
ALDH1A1 P00352 5/20 0.48
NPSR1 Q6W5P4 3/20 0.48
ATM Q13315 2/20 0.48
JAK2 O60674 2/20 0.48
HPGD P15428 2/20 0.48
HTT P42858 2/20 0.48
TP53 P04637 1/20 0.48
MAPK1 P28482 1/20 0.48
HSD17B10 Q99714 1/20 0.48
KLK5 Q9Y337 2/20 0.43
TSHR P16473 3/20 0.43
POLB P06746 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
LMNA P02545 3/20 0.42
PPARG P37231 1/20 0.42
NCOA2 Q15596 1/20 0.42
NCOA1 Q15788 1/20 0.42
NCOA3 Q9Y6Q9 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8892245 1.00 CTSS (0.49) CTSSCTSKALDH1A1NPSR1ATM
SCHEMBL7435053 0.92 CTSS (0.45) CTSSCTSKALDH1A1NPSR1ATM
SCHEMBL7435046 0.92 CTSS (0.45) CTSSCTSKALDH1A1NPSR1ATM
SCHEMBL7283432 0.92 KLK5 (0.47) CTSSCTSKALDH1A1NPSR1ATM
SCHEMBL5142842 0.92 KLK5 (0.47) CTSSCTSKALDH1A1NPSR1ATM
SCHEMBL7398818 0.92 KLK5 (0.47) CTSSCTSKALDH1A1NPSR1ATM
SCHEMBL7796450 0.92 KLK5 (0.47) CTSSCTSKALDH1A1NPSR1ATM
SCHEMBL6305846 0.92 KLK5 (0.47) CTSSCTSKALDH1A1NPSR1ATM
SCHEMBL6446803 0.92 KLK5 (0.47) CTSSCTSKALDH1A1NPSR1ATM
SCHEMBL9546500 0.90 NPSR1 (0.47) CTSSCTSKALDH1A1NPSR1ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5643878-A TREATMENT OF RETROVIRAL DISEASES LIKE AIDS CIBA-GEIGY CORPORATION (US) 1997-07-01 US disclosed
WO-1996016980-A1 MORPHOLINOETHYLAMIDE DERIVATIVES NOVARTIS AG (CH) 1996-06-06 WO disclosed
EP-0618222-A2 Dipeptid derivatives of 5-amino-4-hydroxy-hexanoic acid CIBA-GEIGY AG (CH) 1994-10-05 EP disclosed