SCHEMBL8892263

SCHEMBL8892263

COc1ccc(Oc2c(Cl)cc(N)cc2Cl)cc1Cc1ccc(F)cc1

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
THRB P10828 2/20 0.43
RORC P51449 1/20 0.43
THRA P10827 1/20 0.43
HTR2A P28223 9/20 0.42
SLC6A4 P31645 9/20 0.42
KCNH2 Q12809 8/20 0.42
MEN1 O00255 1/20 0.38
MAPT P10636 1/20 0.38
KMT2A Q03164 1/20 0.38
FDFT1 P37268 1/20 0.37
PPARD Q03181 1/20 0.37
PPARA Q07869 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18998446 0.93 THRB (0.40) THRBRORCTHRAHTR2ASLC6A4
SCHEMBL18932876 0.88 THRB (0.45) THRBRORCHTR2ASLC6A4KCNH2
SCHEMBL282344 0.87 THRB (0.59) THRBRORCTHRAHTR2ASLC6A4
SCHEMBL4960799 0.84 THRB (0.46) THRBRORCTHRAHTR2ASLC6A4
SCHEMBL282509 0.83 ATM (0.46) THRBRORCTHRAHTR2ASLC6A4
SCHEMBL8892137 0.83 MAPT (0.43) THRBRORCTHRAHTR2ASLC6A4
SCHEMBL18918559 0.80 THRB (0.48) THRBRORCTHRA
SCHEMBL18932877 0.79 THRB (0.46) THRBRORCTHRAHTR2ASLC6A4
SCHEMBL3152794 0.79 THRA (0.43) THRBTHRAHTR2AMEN1KMT2A
SCHEMBL18932875 0.77 THRB (0.55) THRBRORCTHRAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3181556-B1 MICROMOLECULE COMPOUND, METHOD OF SYNTHESIS AND APPLICATION THEREOF TECHNODERMA MEDICINES PTE LTD (CN) 2021-09-29 EP disclosed
EP-3181556-B1 MICROMOLECULE COMPOUND, METHOD OF SYNTHESIS AND APPLICATION THEREOF TECHNODERMA MEDICINES PTE LTD (CN) 2021-09-29 EP disclosed
US-9920022-B2 Small molecule compound and synthesizing method and uses thereof TECHNODERMA MEDICINES PTE LTD. (CN) 2018-03-20 US disclosed
US-9920022-B2 Small molecule compound and synthesizing method and uses thereof TECHNODERMA MEDICINES PTE LTD. (CN) 2018-03-20 US disclosed
US-9920022-B2 Small molecule compound and synthesizing method and uses thereof TECHNODERMA MEDICINES PTE LTD. (CN) 2018-03-20 US disclosed
EP-3181556-A1 MICROMOLECULE COMPOUND, METHOD OF SYNTHESIS AND APPLICATION THEREOF Technoderma Medicines Pte Ltd (CN) 2017-06-21 EP disclosed
EP-3181556-A1 MICROMOLECULE COMPOUND, METHOD OF SYNTHESIS AND APPLICATION THEREOF Technoderma Medicines Pte Ltd (CN) 2017-06-21 EP disclosed
US-20170158651-A1 SMALL MOLECULE COMPOUND AND SYNTHESIZING METHOD AND USES THEREOF TECHNODERMA MEDICINES PTE LTD. 2017-06-08 US disclosed
US-20170158651-A1 SMALL MOLECULE COMPOUND AND SYNTHESIZING METHOD AND USES THEREOF TECHNODERMA MEDICINES PTE LTD. 2017-06-08 US disclosed
US-20170158651-A1 SMALL MOLECULE COMPOUND AND SYNTHESIZING METHOD AND USES THEREOF TECHNODERMA MEDICINES PTE LTD. 2017-06-08 US disclosed
US-5654468-A ANTILIPID, ANTICHOLESTEROL AGENTS CIBA-GEIGY CORPORATION (US) 1997-08-05 US disclosed
US-5569674-A ANTICHOLESTEROL AGENTS CIBA-GEIGY CORPORATION (US) 1996-10-29 US disclosed
US-5401772-A Anticholesterol agents with aromatic amines CIBA-GEIGY CORPORATION (US) 1995-03-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170158651-A1 SMALL MOLECULE COMPOUND AND SYNTHESIZING METHOD AND USES THEREOF MKI67, ACP1, TYR THRB 2396/4885RORC 2654/4885THRA 3476/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.