SCHEMBL8892830

SCHEMBL8892830

Cc1cc(N(C)c2ccccc2)cc(=O)n1C

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.54
MAPT P10636 4/20 0.41
LMNA P02545 3/20 0.41
HPGD P15428 3/20 0.41
ALOX15 P16050 1/20 0.41
TSHR P16473 1/20 0.41
KDM4C Q9H3R0 1/20 0.40
KDM4E B2RXH2 1/20 0.39
NQO2 P16083 1/20 0.39
NAPRT Q6XQN6 1/20 0.39
PKM P14618 1/20 0.38
KMT2A Q03164 6/20 0.38
CYP1A2 P05177 3/20 0.38
CYP2C9 P11712 2/20 0.38
CYP2C19 P33261 1/20 0.38
SMN1; SMN2 Q16637 3/20 0.37
MEN1 O00255 3/20 0.37
ALDH1A1 P00352 2/20 0.37
S1PR4 O95977 1/20 0.37
HSP90AA1 P07900 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8895981 0.79 KDM4C (0.57) GAAMAPTLMNAHPGDTSHR
Hydrochloric Acid SCHEMBL8894684 0.78 KDM4C (0.56) GAAMAPTLMNAHPGDTSHR
SCHEMBL8893397 0.73 KDM4C (0.42) GAAMAPTLMNAHPGDALOX15
SCHEMBL12258324 0.72 CHKA (0.47) GAALMNAHPGDKMT2ASMN1; SMN2
SCHEMBL12441468 0.71 HSD17B10 (0.47) MAPTLMNAHPGDKDM4ENQO2
SCHEMBL5307352 0.70 GAA (1.00) GAAMAPTLMNAHPGDALOX15
SCHEMBL20385081 0.69 MEN1 (0.52) LMNAHPGDKMT2ASMN1; SMN2MEN1
SCHEMBL22931682 0.69 MEN1 (0.52) LMNAHPGDKMT2ASMN1; SMN2MEN1
SCHEMBL31886 0.69 MEN1 (0.52) LMNAHPGDKMT2ASMN1; SMN2MEN1
SCHEMBL6567354 0.69 MEN1 (0.52) LMNAHPGDKMT2ASMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5654298-A QUARTERNARY SALTS OF 4-AMINO-SUBSTITUTED PYRIDINES; MODULATORS OF THE SINOATRIAL NODE; CARDIOTONIC AND BRADYCARDIA AGENTS; IMPERIAL CHEMICAL INDUSTRIES (GB) 1997-08-05 US disclosed
EP-0453197-B1 Amine derivatives ICI PLC (GB) 1994-06-15 EP disclosed
EP-0453197-A1 Amine derivatives IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1991-10-23 EP disclosed