SCHEMBL8893397

SCHEMBL8893397

CC#CCN(c1ccccc1)c1cc(C)n(C)c(=O)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4C Q9H3R0 1/20 0.42
KMT2A Q03164 4/20 0.39
SMN1; SMN2 Q16637 4/20 0.39
MEN1 O00255 2/20 0.39
HSD17B10 Q99714 2/20 0.39
CASP1 P29466 1/20 0.39
BRCA1 P38398 1/20 0.39
CASP7 P55210 1/20 0.39
GAA P10253 1/20 0.36
MAPT P10636 3/20 0.32
CYP1A2 P05177 2/20 0.32
HPGD P15428 2/20 0.32
LMNA P02545 2/20 0.32
CYP2C19 P33261 1/20 0.32
CYP2C9 P11712 1/20 0.32
KDM4E B2RXH2 2/20 0.32
NQO2 P16083 1/20 0.32
NAPRT Q6XQN6 1/20 0.32
ALDH1A1 P00352 2/20 0.31
CYP3A4 P08684 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8895981 0.81 KDM4C (0.57) KDM4CKMT2ASMN1; SMN2MEN1HSD17B10
Hydrochloric Acid SCHEMBL8894684 0.80 KDM4C (0.56) KDM4CKMT2ASMN1; SMN2MEN1HSD17B10
SCHEMBL14288498 0.77 MAPT (0.37) KMT2AMEN1GAAMAPTCYP1A2
SCHEMBL22870227 0.75 MAPT (0.37) KMT2AMEN1GAAMAPTCYP1A2
SCHEMBL8892830 0.73 GAA (0.54) KDM4CKMT2ASMN1; SMN2MEN1HSD17B10
SCHEMBL9731530 0.66 KCNH2 (0.38) KMT2AMEN1GAAMAPTCYP1A2
SCHEMBL8894176 0.66 POLB (0.46) KDM4CKMT2ASMN1; SMN2MEN1HSD17B10
SCHEMBL9378372 0.66 HCN1 (0.46) CYP1A2
Hydrochloric Acid SCHEMBL8892491 0.65 POLB (0.45) KDM4CKMT2ASMN1; SMN2MEN1HSD17B10
SCHEMBL8893610 0.65 KDM4C (0.45) KDM4CKMT2ASMN1; SMN2MEN1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5654298-A QUARTERNARY SALTS OF 4-AMINO-SUBSTITUTED PYRIDINES; MODULATORS OF THE SINOATRIAL NODE; CARDIOTONIC AND BRADYCARDIA AGENTS; IMPERIAL CHEMICAL INDUSTRIES (GB) 1997-08-05 US disclosed
EP-0453197-B1 Amine derivatives ICI PLC (GB) 1994-06-15 EP disclosed
EP-0453197-A1 Amine derivatives IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1991-10-23 EP disclosed