SCHEMBL8892980

SCHEMBL8892980

Fc1ccc(C(OCCN2C=CC=NC2)c2ccc(F)cc2)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 3/20 0.49
SLC6A4 P31645 8/20 0.47
SLC6A3 Q01959 8/20 0.47
SLC6A2 P23975 5/20 0.47
LMNA P02545 2/20 0.46
NPSR1 Q6W5P4 1/20 0.46
DRD2 P14416 1/20 0.44
DRD4 P21917 1/20 0.44
DRD3 P35462 1/20 0.44
MEN1 O00255 1/20 0.44
NPC1 O15118 1/20 0.44
ALDH1A1 P00352 1/20 0.44
TP53 P04637 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
MAPT P10636 1/20 0.44
CYP2C9 P11712 1/20 0.44
TSHR P16473 1/20 0.44
NFKB1 P19838 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8892879 0.82 SLC6A3 (0.33) SIGMAR1SLC6A4SLC6A3SLC6A2LMNA
SCHEMBL8892302 0.78 SIGMAR1 (0.51) SIGMAR1SLC6A4SLC6A3SLC6A2LMNA
SCHEMBL8892976 0.70 SIGMAR1 (0.49) SIGMAR1SLC6A4SLC6A3SLC6A2LMNA
SCHEMBL8643721 0.69 SIGMAR1 (0.66) SIGMAR1SLC6A4SLC6A3SLC6A2LMNA
SCHEMBL8642037 0.69 LMNA (0.78) SIGMAR1SLC6A4SLC6A3SLC6A2LMNA
SCHEMBL8647649 0.69 LMNA (0.83) SIGMAR1SLC6A4SLC6A3SLC6A2LMNA
SCHEMBL8645362 0.68 LMNA (0.81) SIGMAR1SLC6A4SLC6A3SLC6A2LMNA
SCHEMBL10551886 0.68 SIGMAR1 (0.73) SIGMAR1SLC6A4SLC6A3SLC6A2LMNA
SCHEMBL9430393 0.68 SIGMAR1 (0.73) SIGMAR1SLC6A4SLC6A3SLC6A2LMNA
SCHEMBL8892780 0.67 SIGMAR1 (0.55) SIGMAR1SLC6A4SLC6A3SLC6A2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997027175-A1 SUBSTITUTED ETHYL α,α - DIARYLMETHYL ETHER DERIVATIVES GUILFORD PHARMACEUTICALS INC. (US) 1997-07-31 WO claimed
WO-1997027175-A1 SUBSTITUTED ETHYL α,α - DIARYLMETHYL ETHER DERIVATIVES GUILFORD PHARMACEUTICALS INC. (US) 1997-07-31 WO disclosed