SCHEMBL8893210

SCHEMBL8893210

COc1ccc(NC2(C(N)=O)CCN(Cc3ccccc3)CC2)cc1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.61
CYP2D6 P10635 2/20 0.61
TSHR P16473 1/20 0.56
SIGMAR1 Q99720 2/20 0.54
NPFFR1 Q9GZQ6 3/20 0.54
NPFFR2 Q9Y5X5 3/20 0.54
OPRM1 P35372 2/20 0.54
OPRK1 P41145 2/20 0.54
MMP1 P03956 2/20 0.54
MMP9 P14780 2/20 0.54
MMP13 P45452 2/20 0.54
ADAM17 P78536 2/20 0.54
OPRD1 P41143 1/20 0.54
FAAH O00519 2/20 0.53
MAPT P10636 1/20 0.53
L3MBTL1 Q9Y468 1/20 0.53
KMT2A Q03164 2/20 0.52
MEN1 O00255 1/20 0.52
POLB P06746 1/20 0.52
ACHE P22303 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11568366 0.91 CYP2D6 (0.58) ALDH1A1CYP2D6TSHRSIGMAR1NPFFR1
SCHEMBL11559495 0.90 CYP2D6 (0.57) ALDH1A1CYP2D6TSHRSIGMAR1NPFFR1
SCHEMBL11564966 0.88 NPFFR1 (0.64) ALDH1A1CYP2D6TSHRSIGMAR1NPFFR1
SCHEMBL13422580 0.88 FAAH (0.61) ALDH1A1CYP2D6SIGMAR1NPFFR1NPFFR2
SCHEMBL2996293 0.88 CYP2D6 (0.68) ALDH1A1CYP2D6TSHRNPFFR1NPFFR2
SCHEMBL3939085 0.87 CYP2D6 (0.65) ALDH1A1CYP2D6TSHRNPFFR1NPFFR2
SCHEMBL654357 0.86 ALDH1A1 (0.62) ALDH1A1CYP2D6TSHRSIGMAR1NPFFR1
SCHEMBL16876712 0.86 ALDH1A1 (0.57) ALDH1A1CYP2D6TSHRNPFFR1NPFFR2
SCHEMBL5556286 0.85 ALDH1A1 (0.61) ALDH1A1CYP2D6TSHRSIGMAR1NPFFR1
SCHEMBL16876726 0.85 ALDH1A1 (0.61) ALDH1A1CYP2D6TSHRSIGMAR1NPFFR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5610142-A Bradykinin antagonist pseudopeptide derivatives of substituted 4-keto-1,3,8-triazaspiro[4.5]decan-3-alkanoic acids SCIOS INC. (US) 1997-03-11 US disclosed