SCHEMBL8893391

SCHEMBL8893391

COc1ccc(N(C(=O)Cl)c2ccccn2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.50
NPC1 O15118 4/20 0.49
RAB9A P51151 4/20 0.49
SMN1; SMN2 Q16637 3/20 0.49
PKM P14618 3/20 0.49
MAPT P10636 3/20 0.49
TRPM8 Q7Z2W7 5/20 0.48
HPGD P15428 1/20 0.47
CDK5 Q00535 1/20 0.47
PAX8 Q06710 1/20 0.47
CDK5R1 Q15078 1/20 0.47
F2 P00734 1/20 0.45
POLB P06746 2/20 0.45
BLM P54132 1/20 0.45
PMP22 Q01453 1/20 0.45
KMT2A Q03164 3/20 0.44
MEN1 O00255 2/20 0.44
ALDH1A1 P00352 2/20 0.44
LMNA P02545 1/20 0.44
CYP1A2 P05177 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7968757 0.87 POLB (0.52) KDM4ENPC1RAB9ASMN1; SMN2PKM
SCHEMBL3906341 0.86 KDM4E (0.51) KDM4ENPC1RAB9ASMN1; SMN2PKM
SCHEMBL1118771 0.80 TRPM8 (0.56) KDM4ETRPM8HPGDPOLBKMT2A
SCHEMBL11540415 0.79 CES2 (0.48) KDM4ENPC1RAB9ASMN1; SMN2MAPT
SCHEMBL12669562 0.77 KDM4E (0.55) KDM4ENPC1RAB9ASMN1; SMN2PKM
SCHEMBL13367406 0.75 MEN1 (0.54) KDM4ENPC1SMN1; SMN2TRPM8BLM
SCHEMBL31098975 0.74 KDM4E (0.52) KDM4ENPC1RAB9ASMN1; SMN2PKM
SCHEMBL7978882 0.72 TP53 (0.49) NPC1RAB9APKMTRPM8CDK5
SCHEMBL13338802 0.72 KDM4E (0.53) KDM4ESMN1; SMN2TRPM8POLBBLM
SCHEMBL20484557 0.72 HTT (0.49) KDM4ENPC1RAB9ASMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997024328-A1 2-AMINO-HETEROCYCLES AND THERAPEUTIC USES THEREFOR BAYER AKTIENGESELLSCHAFT (DE) 1997-07-10 WO disclosed