SCHEMBL8894088

SCHEMBL8894088

Cc1cccc(N2CCCCC2)c1C

nearest known ligand 0.68

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
LMNA P02545 5/20 0.68
MEN1 O00255 3/20 0.68
KMT2A Q03164 3/20 0.68
ADRB1 P08588 1/20 0.67
ALDH1A1 P00352 6/20 0.59
NPSR1 Q6W5P4 2/20 0.59
TSHR P16473 3/20 0.57
MAPK1 P28482 1/20 0.57
MAPT P10636 5/20 0.56
GAA P10253 3/20 0.54
HPGD P15428 2/20 0.54
KDM4E B2RXH2 3/20 0.52
RAB9A P51151 1/20 0.52
ALOX15 P16050 1/20 0.50
HSD17B10 Q99714 1/20 0.50
HSP90AA1 P07900 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
POLB P06746 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9065218 1.00 LMNA (0.68) LMNAMEN1KMT2AADRB1ALDH1A1
SCHEMBL30228454 1.00 LMNA (0.68) LMNAMEN1KMT2AADRB1ALDH1A1
SCHEMBL23843550 0.98 ADRB1 (0.69) LMNAMEN1KMT2AADRB1ALDH1A1
SCHEMBL29058159 0.94 ADRB1 (0.69) LMNAMEN1KMT2AADRB1ALDH1A1
SCHEMBL28762158 0.89 MEN1 (0.61) LMNAMEN1KMT2AADRB1ALDH1A1
SCHEMBL11067105 0.89 ADRB1 (0.74) LMNAMEN1KMT2AADRB1ALDH1A1
SCHEMBL31468714 0.83 ADRB1 (0.64) LMNAMEN1KMT2AADRB1ALDH1A1
SCHEMBL329640 0.83 ADRB1 (0.64) LMNAMEN1KMT2AADRB1ALDH1A1
SCHEMBL2332676 0.83 ADRB1 (0.64) LMNAMEN1KMT2AADRB1ALDH1A1
SCHEMBL329728 0.83 ADRB1 (0.64) LMNAMEN1KMT2AADRB1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023202705-A1 OPHTHALMIC PREPARATION AND APPLICATION THEREOF IN TREATING PRESBYOPIA 温州医科大学附属眼视光医院 2023-10-26 WO disclosed
US-9181245-B2 Substituted pyrido[1,2-a]pyrazines and substituted pyrido[1,2-a][1,4]diazepines for the treatment of (inter alia) Alzheimer's disease Janssen Pharmaceuticals, Inc. (US) 2015-11-10 US disclosed
US-9181245-B2 Substituted pyrido[1,2-a]pyrazines and substituted pyrido[1,2-a][1,4]diazepines for the treatment of (inter alia) Alzheimer's disease Janssen Pharmaceuticals, Inc. (US) 2015-11-10 US disclosed
US-20150141411-A1 SUBSTITUTED 3,4-DIHYDRO-2H-PYRIDO[1,2-A]PYRAZINE-1,6-DIONE DERIVATIVES USEFUL FOR THE TREATMENT OF (INTER ALIA) ALZHEIMER'S DISEASE CELLZOME LIMITED (GB) 2015-05-21 US disclosed
US-20150141411-A1 SUBSTITUTED 3,4-DIHYDRO-2H-PYRIDO[1,2-A]PYRAZINE-1,6-DIONE DERIVATIVES USEFUL FOR THE TREATMENT OF (INTER ALIA) ALZHEIMER'S DISEASE CELLZOME LIMITED (GB) 2015-05-21 US disclosed
CN-100469837-C Fire-retardant resin composition and its molded product GEN ELECTRIC (NL) 2009-03-18 CN disclosed
CN-1234758-C Incombustible resin composition and molded article thereof GEN ELECTRIC (US) 2006-01-04 CN disclosed
CN-1487968-A Flame retardant resin compositon and molded products thereof ͨ�õ�����˾ 2004-04-07 CN disclosed
CN-1370803-A Fire-retardant resin composition and its molded product GEN ELECTRIC (US) 2002-09-25 CN disclosed
WO-1997014689-A1 ARYL-PIPERAZINE CYCLIC AMINE DERIVATIVES, PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME PIERRE FABRE MEDICAMENT (FR) 1997-04-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150141411-A1 SUBSTITUTED 3,4-DIHYDRO-2H-PYRIDO[1,2-A]PYRAZINE-1,6-DIONE DERIVATIVES USEFUL FOR THE TREATMENT OF (INTER ALIA) ALZHEIMER'S DISEASE BACE1, PSEN1, BACE2 LMNA 772/4885MEN1 3484/4885KMT2A 2505/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.