SCHEMBL8894717

SCHEMBL8894717

CC(=O)OCCCc1cc(C=C2SC(=S)N(C)C2=O)cc(CCCOC(C)=O)c1O

nearest known ligand 0.56

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NAT1 P18440 2/20 0.56
HSD17B3 P37058 1/20 0.47
CISD1 Q9NZ45 4/20 0.45
MAOB P27338 2/20 0.45
MAOA P21397 1/20 0.45
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
MAPT P10636 1/20 0.43
CGAS Q8N884 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9027978 1.00 NAT1 (0.56) NAT1HSD17B3CISD1MAOBMAOA
SCHEMBL8896050 0.80 TNKS2 (0.38) NAT1MEN1KMT2A
SCHEMBL8893765 0.75 TNKS2 (0.36)
SCHEMBL9684884 0.74 TNKS2 (0.39) NAT1CISD1MAOBMAOAMEN1
SCHEMBL9684891 0.74 TNKS2 (0.39) NAT1CISD1MAOBMAOAMEN1
SCHEMBL8536492 0.72 NAT1 (0.69) NAT1HSD17B3CISD1MAOBMAOA
SCHEMBL8933387 0.72 HSD17B3 (0.49) NAT1HSD17B3CISD1MAOAMEN1
SCHEMBL8893373 0.72 HSD17B3 (0.49) NAT1HSD17B3CISD1MAOAMEN1
SCHEMBL8198993 0.69 NAT1 (0.69) NAT1HSD17B3CISD1MAOBMAOA
SCHEMBL7246589 0.69 NAT1 (0.69) NAT1HSD17B3CISD1MAOBMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5691367-A ANTIINFLAMMATORY AGENTS OR ANTIARTHRITIC AGENTS ELI LILLY AND COMPANY (US) 1997-11-25 US disclosed
EP-0391644-B1 Aryl-substituted rhodanine derivatives LILLY CO ELI (US) 1996-06-19 EP disclosed
US-5356917-A Antiischemic, antiinflammatory, antiarthritic agents, treat-ment of dystrophic mammals ELI LILLY AND COMPANY (US) 1994-10-18 US disclosed
US-5158966-A Aryl-substituted rhodanine derivatives THE UNIVERSITY OF COLORADO FOUNDATION, INC. (US) 1992-10-27 US disclosed
EP-0391644-A2 Aryl-substituted rhodanine derivatives ELI LILLY AND COMPANY (US) 1990-10-10 EP disclosed