SCHEMBL8893765

SCHEMBL8893765

CC(=O)OCCCc1cc(C=C2SCN(N(C)C)C2=O)cc(CCCOC(C)=O)c1O

nearest known ligand 0.36

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TNKS2 Q9H2K2 1/20 0.36
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2C9 P11712 1/20 0.30
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8896050 0.86 TNKS2 (0.38) TNKS2CYP1A2CYP3A4CYP2C9ALDH1A1
SCHEMBL9684891 0.77 TNKS2 (0.39) TNKS2CYP1A2CYP3A4CYP2C9ALDH1A1
SCHEMBL9684884 0.77 TNKS2 (0.39) TNKS2CYP1A2CYP3A4CYP2C9ALDH1A1
SCHEMBL9027978 0.75 NAT1 (0.56)
SCHEMBL8894717 0.75 NAT1 (0.56)
SCHEMBL8894724 0.68 PTGS2 (0.45) CYP1A2CYP2C9ALDH1A1
SCHEMBL8532254 0.67 CYP1A2 (0.40) CYP1A2CYP3A4CYP2C9ALDH1A1
SCHEMBL8532250 0.67 CYP1A2 (0.40) CYP1A2CYP3A4CYP2C9ALDH1A1
SCHEMBL8991927 0.67 PTGS2 (0.45) CYP1A2CYP2C9ALDH1A1
SCHEMBL8894493 0.67 PTGS2 (0.45) CYP1A2CYP2C9ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5691367-A ANTIINFLAMMATORY AGENTS OR ANTIARTHRITIC AGENTS ELI LILLY AND COMPANY (US) 1997-11-25 US disclosed
EP-0391644-B1 Aryl-substituted rhodanine derivatives LILLY CO ELI (US) 1996-06-19 EP disclosed
US-5356917-A Antiischemic, antiinflammatory, antiarthritic agents, treat-ment of dystrophic mammals ELI LILLY AND COMPANY (US) 1994-10-18 US disclosed
EP-0391644-A2 Aryl-substituted rhodanine derivatives ELI LILLY AND COMPANY (US) 1990-10-10 EP disclosed