SCHEMBL8895514

SCHEMBL8895514

COC(=O)CCC1CCC(NC(=O)N(CC(=O)OCc2ccccc2)c2ccc3c(c2)CCN(C(=O)C(F)(F)F)CC3)CC1

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 11/20 0.37
ESR1 P03372 1/20 0.36
ESR2 Q92731 1/20 0.36
DRD3 P35462 2/20 0.36
TMEM97 Q5BJF2 2/20 0.35
SIGMAR1 Q99720 2/20 0.35
HTT P42858 1/20 0.35
GPR183 P32249 1/20 0.34
CHRM4 P08173 1/20 0.34
MEN1 O00255 1/20 0.34
ALDH1A1 P00352 1/20 0.34
CYP3A4 P08684 1/20 0.34
TSHR P16473 1/20 0.34
MAPK1 P28482 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8895505 1.00 DRD2 (0.37) DRD2ESR1ESR2DRD3TMEM97
SCHEMBL8897546 0.82 ESR1 (0.38) DRD2ESR1ESR2DRD3
SCHEMBL8897540 0.82 ESR1 (0.38) DRD2ESR1ESR2DRD3
SCHEMBL8565938 0.81 TMEM97 (0.37) ESR1ESR2DRD3TMEM97SIGMAR1
SCHEMBL8562609 0.69 ESR1 (0.44) ESR1ESR2DRD3TMEM97SIGMAR1
SCHEMBL7423187 0.68 ESR1 (0.39) ESR1ESR2
SCHEMBL8565611 0.68 DCUN1D1 (0.39) ESR1ESR2MEN1KMT2A
SCHEMBL8565613 0.68 DCUN1D1 (0.39) ESR1ESR2MEN1KMT2A
SCHEMBL8896148 0.67 MCHR1 (0.41)
SCHEMBL8896160 0.67 MCHR1 (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5612335-A ANTICOAGULANTS; COMBATING/PREVENTING DISEASES WHERE CELL AGGREGATES OCCUR OR CELL-MATRIX INTERACTIONS PLAY A PART KARL THOMAE GMBH (DE) 1997-03-18 US disclosed
US-5519036-A IMIDAZOLIDINONES, ANTICOAGULANTS, CELL AGGREGATION PREVENTION KARL THOMAE GMBH (DE) 1996-05-21 US disclosed