SCHEMBL8895567

SCHEMBL8895567

COC(=O)CCCc1ccc(C(N)Cc2ccccc2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C19 P33261 1/20 0.47
KMT2A Q03164 3/20 0.45
ALDH1A1 P00352 2/20 0.45
CA12 O43570 1/20 0.45
CA7 P43166 1/20 0.45
CA9 Q16790 1/20 0.45
CA14 Q9ULX7 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
HDAC1 Q13547 2/20 0.44
ADRB2 P07550 1/20 0.44
ADRB1 P08588 1/20 0.44
ADRB3 P13945 1/20 0.44
RECQL P46063 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
HDAC3 O15379 1/20 0.44
MAPK1 P28482 1/20 0.44
ADRA1A P35348 1/20 0.44
HDAC4 P56524 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8894974 0.86 ADRB3 (0.49) KMT2AALDH1A1CA12CA7CA9
SCHEMBL8896262 0.84 ALDH1A1 (0.45) KMT2AALDH1A1CA12CA7CA9
SCHEMBL7037486 0.83 SLC7A5 (0.55) CYP1A2CYP2D6CYP2C19KMT2AALDH1A1
SCHEMBL162806 0.83 HDAC1 (0.62) KMT2AALDH1A1CA12CA7CA9
SCHEMBL9231232 0.83 ADRB3 (0.47) CA12CA7CA9CA14HDAC1
SCHEMBL9231881 0.81 HDAC1 (0.60) ALDH1A1CA12CA7CA9CA14
Phosphine SCHEMBL27480219 0.81 HDAC1 (0.60) KMT2AALDH1A1CA12CA7CA9
SCHEMBL9233223 0.80 FAAH (0.49) KMT2AALDH1A1CA12CA7CA9
SCHEMBL9235461 0.79 FAAH (0.51) KMT2AALDH1A1HDAC1ADRB2ADRB1
SCHEMBL8894908 0.78 CA12 (0.45) KMT2AALDH1A1CA12CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5597848-A PLATELET AGGREGATION INHIBITORS, ANTITHROMBOTIC AGENTS, ANTIASTHMATIC AGENTS, ANTIALLERGIC AGENTS HOKURIKU SEIYAKU CO., LTD. (JP) 1997-01-28 US disclosed
EP-0663392-A1 BENZENESULFONAMIDE DERIVATIVE AND USE THEREOF HOKURIKU SEIYAKU CO., LTD. (JP) 1995-07-19 EP disclosed