SCHEMBL8895912

SCHEMBL8895912

COc1ccc(C[C@H](N)[C@@H](O)C[C@@H](Cc2ccccc2OC)C(=O)O)cc1

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.50
CYP2C9 P11712 1/20 0.50
LDHA P00338 1/20 0.46
PPARA Q07869 4/20 0.44
PPARG P37231 3/20 0.43
LTA4H P09960 1/20 0.42
MMP1 P03956 2/20 0.42
SLC1A5 Q15758 1/20 0.42
ANPEP P15144 1/20 0.42
ERAP2 Q6P179 1/20 0.42
ALDH1A1 P00352 1/20 0.42
GAA P10253 1/20 0.42
PPARD Q03181 2/20 0.41
REN P00797 1/20 0.41
SLC1A3 P43003 1/20 0.41
SLC1A2 P43004 1/20 0.41
SLC1A1 P43005 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8895907 1.00 CYP1A2 (0.50) CYP1A2CYP2C9LDHAPPARAPPARG
SCHEMBL8894728 0.93 SLC1A3 (0.48) CYP1A2CYP2C9PPARAANPEPALDH1A1
SCHEMBL8894736 0.93 SLC1A3 (0.48) CYP1A2CYP2C9PPARAANPEPALDH1A1
SCHEMBL8893679 0.88 SLC1A3 (0.54) CYP1A2LDHAPPARAPPARGLTA4H
SCHEMBL7439274 0.88 SLC1A3 (0.54) CYP1A2LDHAPPARAPPARGLTA4H
SCHEMBL7439269 0.88 SLC1A3 (0.54) CYP1A2LDHAPPARAPPARGLTA4H
SCHEMBL8893674 0.88 SLC1A3 (0.54) CYP1A2LDHAPPARAPPARGLTA4H
SCHEMBL8891774 0.87 LDHA (0.56) CYP1A2LDHAPPARAPPARGLTA4H
SCHEMBL8891766 0.87 LDHA (0.56) CYP1A2LDHAPPARAPPARGLTA4H
SCHEMBL8892836 0.82 LDHA (0.51) LDHAPPARAPPARGLTA4HMMP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5643878-A TREATMENT OF RETROVIRAL DISEASES LIKE AIDS CIBA-GEIGY CORPORATION (US) 1997-07-01 US disclosed
EP-0618222-A2 Dipeptid derivatives of 5-amino-4-hydroxy-hexanoic acid CIBA-GEIGY AG (CH) 1994-10-05 EP disclosed