SCHEMBL8896337

SCHEMBL8896337

COC(=O)CCCc1ccc(C(CCc2ccccc2)NS(=O)(=O)c2ccc(F)cc2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.45
ATM Q13315 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
POLB P06746 1/20 0.45
MMP2 P08253 2/20 0.43
MMP9 P14780 2/20 0.43
MMP8 P22894 2/20 0.43
MMP14 P50281 2/20 0.43
MMP12 P39900 1/20 0.43
LMNA P02545 1/20 0.43
TAAR1 Q96RJ0 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
EEF2K O00418 1/20 0.41
CA12 O43570 1/20 0.41
CA7 P43166 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8896413 0.92 ALDH1A1 (0.45) ALDH1A1ATML3MBTL1MMP2MMP9
SCHEMBL8895038 0.91 UTS2R (0.45) ALDH1A1LMNACYP1A2CYP2C9CYP2C19
SCHEMBL8897043 0.90 ALDH1A1 (0.46) ALDH1A1ATML3MBTL1POLBMMP2
SCHEMBL8895380 0.90 IDO1 (0.50) ALDH1A1ATML3MBTL1POLBMMP2
SCHEMBL8898350 0.90 ALDH1A1 (0.48) ALDH1A1ATML3MBTL1MMP2MMP9
SCHEMBL8894981 0.89 FFAR1 (0.48) ALDH1A1ATML3MBTL1POLBMMP2
SCHEMBL8897514 0.89 NPSR1 (0.42) ALDH1A1ATML3MBTL1POLBMMP2
SCHEMBL8896101 0.88 FFAR1 (0.47) ALDH1A1ATML3MBTL1POLBLMNA
SCHEMBL8895376 0.88 SIGMAR1 (0.41) ALDH1A1ATML3MBTL1POLBMMP2
SCHEMBL8895525 0.88 SIGMAR1 (0.41) ALDH1A1ATML3MBTL1POLBMMP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5597848-A PLATELET AGGREGATION INHIBITORS, ANTITHROMBOTIC AGENTS, ANTIASTHMATIC AGENTS, ANTIALLERGIC AGENTS HOKURIKU SEIYAKU CO., LTD. (JP) 1997-01-28 US disclosed
EP-0663392-A1 BENZENESULFONAMIDE DERIVATIVE AND USE THEREOF HOKURIKU SEIYAKU CO., LTD. (JP) 1995-07-19 EP disclosed