SCHEMBL8896473

SCHEMBL8896473

O=C(CCCN1CN(c2ccccc2)C2(CCNCC2)C1=O)c1ccc(F)cc1

nearest known ligand 0.72

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.65
DRD4 P21917 1/20 0.65
HTR2A P28223 1/20 0.65
DRD3 P35462 1/20 0.65
MEN1 O00255 1/20 0.63
TP53 P04637 1/20 0.63
CYP1A2 P05177 1/20 0.63
CYP3A4 P08684 1/20 0.63
CYP2D6 P10635 1/20 0.63
MAPT P10636 1/20 0.63
ALOX15 P16050 1/20 0.63
TSHR P16473 1/20 0.63
MAPK1 P28482 1/20 0.63
CYP2C19 P33261 1/20 0.63
KMT2A Q03164 1/20 0.63
SMN1; SMN2 Q16637 1/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29462918 0.83 DRD2 (0.79) DRD2DRD4HTR2ADRD3MEN1
Hydrochloric Acid SCHEMBL30050104 0.82 DRD2 (0.76) DRD2DRD4HTR2ADRD3MEN1
SCHEMBL5108598 0.81 OPRL1 (0.52)
SCHEMBL318863 0.79 OPRL1 (0.49)
Mespiperone SCHEMBL1901596 0.79 DRD2 (1.00) DRD2DRD4HTR2ADRD3MEN1
SCHEMBL30405289 0.79 DRD2 (0.74) DRD2DRD4HTR2ADRD3MEN1
Mespiperone SCHEMBL10733631 0.78 DRD2 (0.98) DRD2DRD4HTR2ADRD3MEN1
SCHEMBL319140 0.78 BDKRB2 (0.49) MEN1CYP3A4CYP2D6KMT2A
SCHEMBL29430174 0.77 MEN1 (1.00) DRD2DRD4HTR2ADRD3MEN1
SCHEMBL13073119 0.77 MEN1 (1.00) DRD2DRD4HTR2ADRD3MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5703088-A Topical application of spiperone or derivatives thereof for treatment of pathological conditions associated with immune responses BETH ISRAEL DEACONESS MEDICAL CENTER, INC. (US) 1997-12-30 US disclosed
US-5693645-A TOPICALLY OR SYSTEMICALLY ADMINISTERING TO THE MAMMAL; USEFUL FOR TREATING INFLAMMATORY BOWL DISEASE BETH ISRAEL DEACONESS MEDICAL CENTER, INC. (US) 1997-12-02 US disclosed