SCHEMBL8896716

SCHEMBL8896716

CC1C=C2c3cc(Br)ccc3C(C)(C)CC21

nearest known ligand 0.35

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 1/20 0.35
PBRM1 Q86U86 1/20 0.31
TDP2 O95551 1/20 0.30
ADRA2A P08913 1/20 0.30
PNMT P11086 1/20 0.30
ADRA2B P18089 1/20 0.30
ADRA2C P18825 1/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8563483 0.72 RXRA (0.32)
SCHEMBL6814457 0.72 PBRM1 (0.39) PDE4BPBRM1TDP2MEN1KMT2A
SCHEMBL6878453 0.69 ESR2 (0.43) PDE4BPBRM1TDP2MEN1KMT2A
SCHEMBL24806899 0.66 KDM1A (0.37) PDE4BADRA2APNMTADRA2BADRA2C
SCHEMBL24806881 0.66 KDM1A (0.37) PDE4BADRA2APNMTADRA2BADRA2C
SCHEMBL6876533 0.66 PDE4B (0.34) PDE4BPBRM1TDP2MEN1KMT2A
SCHEMBL7880635 0.64 PDE4B (0.46) PDE4BTDP2MEN1KMT2A
SCHEMBL484599 0.64 PDE4B (0.46) PDE4BPBRM1TDP2MEN1KMT2A
SCHEMBL6280501 0.63 BACE1 (0.33) PDE4BPBRM1TDP2ADRA2APNMT
SCHEMBL8026081 0.62 ALDH1A1 (0.38) ADRA2APNMTADRA2BADRA2CMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997048672-A2 SUBSTITUTED TETRAHYDRONAPHTHALENE AND DIHYDRONAPHTHALENE DERIVATIVES HAVING RETINOID AND/OR RETINOID ANTAGONIST-LIKE BIOLOGICAL ACTIVITY ALLERGAN SALES, INC. (US) 1997-12-24 WO disclosed