SCHEMBL8897619

SCHEMBL8897619

COC(=O)CCCc1ccc(C(Cc2ccc(C)cc2)NS(=O)(=O)c2ccc(Br)cc2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.50
EGFR P00533 1/20 0.45
ERBB2 P04626 1/20 0.45
RAB9A P51151 1/20 0.42
TDP1 Q9NUW8 2/20 0.42
KDM4E B2RXH2 1/20 0.42
POLB P06746 1/20 0.42
APEX1 P27695 1/20 0.42
RECQL P46063 1/20 0.42
ALDH1A1 P00352 4/20 0.42
CYP3A4 P08684 1/20 0.41
CYP2C19 P33261 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
MMP2 P08253 2/20 0.40
LMNA P02545 1/20 0.40
MMP1 P03956 1/20 0.40
MMP3 P08254 1/20 0.40
MMP7 P09237 1/20 0.40
MMP9 P14780 1/20 0.40
MMP13 P45452 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8895500 0.92 IDO1 (0.50) IDO1RAB9ATDP1POLBALDH1A1
SCHEMBL8895679 0.91 IDO1 (0.49) IDO1EGFRERBB2RAB9APOLB
SCHEMBL8896324 0.91 IDO1 (0.49) IDO1EGFRERBB2RAB9ATDP1
SCHEMBL8894878 0.91 IDO1 (0.49) IDO1EGFRERBB2RAB9APOLB
SCHEMBL8894760 0.91 ALDH1A1 (0.48) RAB9ATDP1ALDH1A1CYP3A4CYP2C19
SCHEMBL8895989 0.90 UTS2R (0.51) EGFRERBB2TDP1ALDH1A1CYP3A4
SCHEMBL8896200 0.90 EGFR (0.45) EGFRERBB2RAB9ATDP1ALDH1A1
SCHEMBL8896314 0.90 ALDH1A1 (0.51) IDO1EGFRERBB2RAB9ATDP1
SCHEMBL8895603 0.87 IDO1 (0.51) IDO1EGFRERBB2RAB9APOLB
SCHEMBL8895471 0.85 NPSR1 (0.44) IDO1KDM4EALDH1A1CYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5597848-A PLATELET AGGREGATION INHIBITORS, ANTITHROMBOTIC AGENTS, ANTIASTHMATIC AGENTS, ANTIALLERGIC AGENTS HOKURIKU SEIYAKU CO., LTD. (JP) 1997-01-28 US disclosed
EP-0663392-A1 BENZENESULFONAMIDE DERIVATIVE AND USE THEREOF HOKURIKU SEIYAKU CO., LTD. (JP) 1995-07-19 EP disclosed