SCHEMBL8894878

SCHEMBL8894878

COC(=O)CCCc1ccc(C(Cc2ccc(Br)cc2)NS(=O)(=O)c2ccc(Cl)cc2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.49
POLB P06746 1/20 0.44
GRK2 P25098 1/20 0.44
KMT2A Q03164 1/20 0.44
EGFR P00533 2/20 0.44
ERBB2 P04626 2/20 0.44
RAB9A P51151 1/20 0.44
ALDH1A1 P00352 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
TSHR P16473 1/20 0.41
MAPK1 P28482 1/20 0.41
CYP2C19 P33261 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
UTS2R Q9UKP6 1/20 0.41
TBXA2R P21731 1/20 0.41
TBXAS1 P24557 1/20 0.41
S1PR1 P21453 4/20 0.40
HDAC3 O15379 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8895679 1.00 IDO1 (0.49) IDO1POLBGRK2KMT2AEGFR
SCHEMBL8895471 0.95 NPSR1 (0.44) IDO1ALDH1A1CYP1A2CYP3A4CYP2C9
SCHEMBL8895500 0.91 IDO1 (0.50) IDO1POLBRAB9AALDH1A1NPSR1
SCHEMBL8897619 0.91 IDO1 (0.50) IDO1POLBKMT2AEGFRERBB2
SCHEMBL8896474 0.91 ADAMTS5 (0.49) ALDH1A1S1PR1ADAMTS5MMP2
SCHEMBL8895989 0.91 UTS2R (0.51) KMT2AEGFRERBB2ALDH1A1CYP1A2
SCHEMBL8897821 0.90 S1PR1 (0.49) EGFRERBB2ALDH1A1CYP1A2CYP3A4
SCHEMBL8895761 0.90 ALDH1A1 (0.49) POLBKMT2AEGFRERBB2ALDH1A1
SCHEMBL8896968 0.90 S1PR1 (0.49) EGFRERBB2ALDH1A1CYP1A2CYP3A4
SCHEMBL8896324 0.90 IDO1 (0.49) IDO1POLBEGFRERBB2RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5597848-A PLATELET AGGREGATION INHIBITORS, ANTITHROMBOTIC AGENTS, ANTIASTHMATIC AGENTS, ANTIALLERGIC AGENTS HOKURIKU SEIYAKU CO., LTD. (JP) 1997-01-28 US disclosed
EP-0663392-A1 BENZENESULFONAMIDE DERIVATIVE AND USE THEREOF HOKURIKU SEIYAKU CO., LTD. (JP) 1995-07-19 EP disclosed