SCHEMBL8897722

SCHEMBL8897722

COc1cnc(C(=O)O)cc1OCc1nc(-c2ccc(Cl)cc2)no1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 1/20 0.54
TSHR P16473 6/20 0.53
MAPK1 P28482 3/20 0.53
TDP1 Q9NUW8 1/20 0.53
THRB P10828 2/20 0.52
GSTP1 P09211 2/20 0.52
MAPT P10636 8/20 0.52
FFAR1 O14842 1/20 0.52
EPHA2 P29317 1/20 0.50
KDR P35968 1/20 0.50
EPHB4 P54760 1/20 0.50
L3MBTL1 Q9Y468 3/20 0.49
LMNA P02545 3/20 0.49
NPC1 O15118 2/20 0.49
RAB9A P51151 2/20 0.49
SMN1; SMN2 Q16637 2/20 0.49
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
TP53 P04637 3/20 0.48
HPGD P15428 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8899814 0.94 SCN9A (0.50) SCN9ATSHRMAPK1TDP1THRB
SCHEMBL8901439 0.91 THRB (0.54) SCN9ATSHRMAPK1TDP1THRB
SCHEMBL8899857 0.85 MAPT (0.58) SCN9ATSHRMAPK1TDP1THRB
SCHEMBL8890864 0.85 THRB (0.51) SCN9ATSHRMAPK1THRBGSTP1
SCHEMBL8892213 0.81 MAPT (0.58) SCN9ATSHRMAPK1TDP1THRB
SCHEMBL8898815 0.77 TSHR (0.59) TSHRMAPK1TDP1THRBGSTP1
SCHEMBL8890753 0.76 MAPT (0.68) TSHRMAPK1THRBGSTP1MAPT
SCHEMBL8890634 0.76 PDE4D (0.60) TSHRMAPK1THRBGSTP1MAPT
SCHEMBL12171456 0.74 MAPT (0.74) TSHRMAPK1TDP1MAPTFFAR1
SCHEMBL8891881 0.72 MAPT (0.49) TSHRMAPK1TDP1THRBGSTP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997003967-A1 SUBSTITUTED AROMATIC COMPOUNDS AND THEIR PHARMACEUTICAL USE RHONE-POULENC RORER LIMITED (GB) 1997-02-06 WO disclosed