SCHEMBL8898613

SCHEMBL8898613

COc1ccc(OC)c(-c2c[nH]c(/N=C/c3ccccc3N)n2)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.41
ALDH1A1 P00352 5/20 0.41
KDM4E B2RXH2 3/20 0.41
NPC1 O15118 3/20 0.41
RAB9A P51151 3/20 0.41
RECQL P46063 2/20 0.41
HPGD P15428 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
GLA P06280 1/20 0.41
GAA P10253 1/20 0.41
L3MBTL1 Q9Y468 2/20 0.38
CYP2C9 P11712 2/20 0.38
CYP2D6 P10635 1/20 0.38
MAPK1 P28482 2/20 0.37
KMT2A Q03164 5/20 0.37
MEN1 O00255 4/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C19 P33261 1/20 0.37
THRB P10828 1/20 0.36
TP53 P04637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8898621 1.00 MAPT (0.41) MAPTALDH1A1KDM4ENPC1RAB9A
SCHEMBL8900342 0.88 HSP90AA1 (0.41) MAPTALDH1A1HPGDGAAALOX15
SCHEMBL8900347 0.88 HSP90AA1 (0.41) MAPTALDH1A1HPGDGAAALOX15
SCHEMBL8899541 0.84 MKNK1 (0.42) MAPTALDH1A1KDM4ERAB9ARECQL
SCHEMBL8899549 0.84 MKNK1 (0.42) MAPTALDH1A1KDM4ERAB9ARECQL
SCHEMBL8898734 0.71 PTGS2 (0.36) MAPTALDH1A1KDM4ENPC1RAB9A
SCHEMBL8898721 0.71 PTGS2 (0.36) MAPTALDH1A1KDM4ENPC1RAB9A
SCHEMBL8900106 0.69 ALDH1A1 (0.32) MAPTALDH1A1KDM4EGAAKMT2A
SCHEMBL8900098 0.69 ALDH1A1 (0.32) MAPTALDH1A1KDM4EGAAKMT2A
SCHEMBL398186 0.67 HDAC4 (0.58) MAPTALDH1A1KDM4ERECQLHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0808309-A1 IMIDAZOLE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS S-ADENOSYLMETHIONINE DECARBOXYLASE (=SAMDC) INHIBITORS Novartis AG (CH) 1997-11-26 EP disclosed
WO-1996022979-A1 IMIDAZOLE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS S-ADENOSYLMETHIONINE DECARBOXYLASE (=SAMDC) INHIBITORS NOVARTIS AG (CH) 1996-08-01 WO disclosed