Bromide

Bromide

SCHEMBL8899853

CC(C)(C)OC(=O)CCC(=O)Nc1ccc(CN2CC[C@@H]([P+](c3ccccc3)(c3ccccc3)c3ccccc3)C2=O)cc1.[Br-]

nearest known ligand 0.41

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHECHKACHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGHRH2OPRM1

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PKM P14618 3/20 0.41
MAPT P10636 4/20 0.41
GAA P10253 3/20 0.41
HDAC8 Q9BY41 3/20 0.37
HDAC3 O15379 1/20 0.37
NCOR2 Q9Y618 1/20 0.37
ALDH1A1 P00352 3/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
KMT2A Q03164 3/20 0.37
MEN1 O00255 2/20 0.37
LTA4H P09960 1/20 0.37
POLB P06746 1/20 0.37
HCRTR1 O43613 1/20 0.37
CCKBR P32239 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL8899846 1.00 PKM (0.41) PKMMAPTGAAHDAC8HDAC3
SCHEMBL8563968 0.81 HDAC8 (0.40) PKMMAPTGAAHDAC8HDAC3
Bromide SCHEMBL8565335 0.81 SIRT2 (0.48) HDAC8HDAC1HDAC6KMT2AMEN1
Bromide SCHEMBL7619361 0.79 PLA2G10 (0.45) PKMMAPTALDH1A1POLBSMN1; SMN2
Bromide SCHEMBL7619358 0.79 PLA2G10 (0.45) PKMMAPTALDH1A1POLBSMN1; SMN2
Bromide SCHEMBL8561888 0.76 TGM2 (0.44) PKMGAAHDAC8ALDH1A1HDAC1
Bromide SCHEMBL8899312 0.76 TGM2 (0.44) PKMGAAHDAC8ALDH1A1HDAC1
Bromide SCHEMBL8563399 0.75 HDAC1 (0.43) HDAC8ALDH1A1HDAC1HDAC6KMT2A
Bromide SCHEMBL8563395 0.75 HDAC1 (0.43) HDAC8ALDH1A1HDAC1HDAC6KMT2A
Bromide SCHEMBL8562995 0.74 MAPT (0.38) MAPTGAAHDAC8ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0761673-A1 Cephalosporin derivatives F. HOFFMANN-LA ROCHE AG (CH) 1997-03-12 EP disclosed