SCHEMBL8563968

SCHEMBL8563968

CC(C)(C)OC(=O)CCC(=O)Nc1ccc(CN2CCC(Br)C2=O)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 3/20 0.40
PKM P14618 2/20 0.40
ALDH1A1 P00352 2/20 0.39
MAPT P10636 2/20 0.39
HDAC3 O15379 1/20 0.39
NCOR2 Q9Y618 1/20 0.39
HPGD P15428 1/20 0.39
FPR2 P25090 1/20 0.39
GAA P10253 3/20 0.39
TSHR P16473 1/20 0.39
HSD17B10 Q99714 1/20 0.39
CACNA1G O43497 1/20 0.39
CHRM1 P11229 1/20 0.39
HTR2A P28223 1/20 0.39
MCHR1 Q99705 1/20 0.39
HDAC1 Q13547 1/20 0.38
HDAC2 Q92769 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
TP53 P04637 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8569448 0.86 DRD2 (0.45) HDAC8ALDH1A1HDAC3NCOR2FPR2
Bromide SCHEMBL8899846 0.81 PKM (0.41) HDAC8PKMALDH1A1MAPTHDAC3
Bromide SCHEMBL8899853 0.81 PKM (0.41) HDAC8PKMALDH1A1MAPTHDAC3
SCHEMBL8561859 0.78 SIRT2 (0.49) HDAC8HDAC1HDAC6TP53
SCHEMBL27520459 0.78 TNIK (0.46) HDAC8PKMALDH1A1FPR2GAA
SCHEMBL8563972 0.73 TP53 (0.37) HDAC1HDAC6TP53
SCHEMBL8560030 0.72 TGM2 (0.46) ALDH1A1MAPTL3MBTL1
SCHEMBL7617920 0.72 PLA2G10 (0.46) ALDH1A1FPR2
SCHEMBL7617915 0.72 PLA2G10 (0.46) ALDH1A1FPR2
SCHEMBL16874550 0.69 KCNH2 (0.51) TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5804577-A ANTIBIOTICS HOFFMANN-LA ROCHE INC. (US) 1998-09-08 US disclosed
EP-0761673-A1 Cephalosporin derivatives F. HOFFMANN-LA ROCHE AG (CH) 1997-03-12 EP disclosed