Lysine

Lysine

SCHEMBL890044

NCCCC[C@@H](N)C(=O)O.N[C@H](CCC(=O)O)C(=O)O

nearest known ligand 0.80

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

PPARDPTGS1PTGS2dacAdacBdacCftsImrcAmrcBmrdA

The experimentally established mechanism targets of Lysine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSR P00390 2/20 0.80
CYP1A2 P05177 2/20 0.72
GRM8 O00222 1/20 0.72
GRM6 O15303 1/20 0.72
GRIN2D O15399 1/20 0.72
GRIN3B O60391 1/20 0.72
GRIK1 P39086 1/20 0.72
GRM5 P41594 1/20 0.72
GRIA1 P42261 1/20 0.72
GRIA2 P42262 1/20 0.72
GRIA3 P42263 1/20 0.72
SLC1A3 P43003 1/20 0.72
SLC1A2 P43004 1/20 0.72
SLC1A1 P43005 1/20 0.72
GRIA4 P48058 1/20 0.72
GRIN1 Q05586 1/20 0.72
GRIN2A Q12879 1/20 0.72
GRIK2 Q13002 1/20 0.72
GRIK3 Q13003 1/20 0.72
GRIN2B Q13224 1/20 0.72

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Lysine SCHEMBL8000337 1.00 GSR (0.80) GSRCYP1A2GRM8GRM6GRIN2D
D-Glutamate SCHEMBL27400214 1.00 GSR (0.80) GSRCYP1A2GRM8GRM6GRIN2D
Lysine SCHEMBL7258645 1.00 GSR (0.80) GSRCYP1A2GRM8GRM6GRIN2D
D-Glutamate SCHEMBL1079951 1.00 GSR (0.80) GSRCYP1A2GRM8GRM6GRIN2D
Lysine SCHEMBL1079952 1.00 GSR (0.80) GSRCYP1A2GRM8GRM6GRIN2D
Lysine SCHEMBL8000334 1.00 GSR (0.80) GSRCYP1A2GRM8GRM6GRIN2D
D-Glutamate SCHEMBL2415481 1.00 GSR (0.80) GSRCYP1A2GRM8GRM6GRIN2D
Lysine SCHEMBL205003 1.00 GSR (0.80) GSRCYP1A2GRM8GRM6GRIN2D
D-Glutamate SCHEMBL21796040 1.00 GSR (0.80) GSRCYP1A2GRM8GRM6GRIN2D
Lysine SCHEMBL6034319 0.98 GSR (0.77) GSRCYP1A2GRM8GRM6GRIN2D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 576 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005040338-A2 CONSTRAINED ALKALOID IMMUNOGENS AND ANTIBODIES AND USES THEREOF THE SCRIPPS RESEARCH INSTITUTE (US) 2005-05-06 WO claimed
US-20240156961-A1 TISSUE-SPECIFIC ANTIGENS FOR CANCER IMMUNOTHERAPY BIONTECH US INC. 2024-05-16 US disclosed
WO-2024077256-A9 METHODS AND COMPOSITIONS FOR HIGH-THROUGHPUT DISCOVERY OF PEPTIDE-MHC TARGETING BINDING PROTEINS THE GENERAL HOSPITAL CORPORATION (US) 2024-05-16 WO disclosed
US-11965892-B2 HLA-based methods and compositions and uses thereof BIONTECH US INC. (US) 2024-04-23 US disclosed
WO-2024081791-A2 COMPOSITIONS AND METHODS FOR MAINTAINING A CCL3/CCL4 AND CCR5 INTERACTION PROGRAM EXPRESSED DURING TUMOR PROGRESSION THE BRIGHAM AND WOMEN'S HOSPITAL, INC. (US) 2024-04-18 WO disclosed
US-20240115678-A1 PERSONALIZED MULTIDISCIPLINARY CANCER THERAPY VELTMEYER JAMES (US) 2024-04-11 US disclosed
WO-2024077256-A1 METHODS AND COMPOSITIONS FOR HIGH-THROUGHPUT DISCOVERY OFPEPTIDE-MHC TARGETING BINDING PROTEINS THE GENERAL HOSPITAL CORPORATION (US) 2024-04-11 WO disclosed
US-20240108690-A1 COMPOSITIONS AND METHODS OF USE OF INTERLEUKIN-10 IN COMBINATION WITH IMMUNE CHECK-POINT PATHWAY INHIBITORS ELI LILLY AND COMPANY 2024-04-04 US disclosed
US-20240100139-A1 NEOANTIGENS AND USES THEREOF BIONTECH US INC. 2024-03-28 US disclosed
US-20240100160-A1 ENHANCEMENT OF T CELL HOMING TO TUMORS THROUGH AUGMENTATION OF CHEMOKINE RESPONSIVENESS AND ACTIVATION DEPENDENT CHEMOKINE SECRETION Regen BioPharma, Inc. (US) 2024-03-28 US disclosed
US-4599231-A MIXTURES OF POLYPOEPTIDES SCRIPPS CLINIC AND RESEARCH FOUNDATION (US) 1986-07-08 US disclosed
US-4599230-A POLYPEPTIDE ANTIGENS SCRIPPS CLINIC AND RESEARCH FOUNDATION (US) 1986-07-08 US disclosed
WO-1985004653-A1 ANTIBODIES TO HUMAN INTERLEUKIN-2 INDUCED BY SYNTHETIC POLYPEPTIDES SCRIPPS CLINIC AND RESEARCH FOUNDATION (US) 1985-10-24 WO disclosed
EP-0157643-A2 Antibodies to human interleukin-2 induced by synthetic polypeptides SCRIPPS CLINIC AND RESEARCH FOUNDATION (US) 1985-10-09 EP disclosed
WO-1985004103-A1 SYNTHETIC HEPATITIS B VIRUS VACCINE INCLUDING BOTH T CELL ANC B CELL DETERMINANTS SCRIPPS CLINIC AND RESEARCH FOUNDATION (US) 1985-09-26 WO disclosed
EP-0155147-A2 The antigenic determinants of HBxAg SCRIPPS CLINIC AND RESEARCH FOUNDATION (US) 1985-09-18 EP disclosed
EP-0155146-A2 Synthetic hepatitis B virus vaccine including both T cell and B cell determinants SCRIPPS CLINIC AND RESEARCH FOUNDATION (US) 1985-09-18 EP disclosed
WO-1985003950-A1 A SV40 EXPRESSION VECTOR CONTAINING HBXAG AS AN EXPRESSION MARKER SCRIPPS CLINIC AND RESEARCH FOUNDATION (US) 1985-09-12 WO disclosed
EP-0119702-A2 Synthetic polypeptides from viral oncogenes Sen, Arup (US) 1984-09-26 EP disclosed
WO-1984003087-A1 SYNTHETIC POLYPEPTIDES FROM VIRAL ONCOGENES SEN ARUP 1984-08-16 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240108690-A1 COMPOSITIONS AND METHODS OF USE OF INTERLEUKIN-10 IN COMBINATION WITH IMMUNE CHECK-POINT PATHWAY INHIBITORS PDCD10, CD274, PDCD1 GSR 4191/4885CYP1A2 4474/4885GRM8 3296/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.