SCHEMBL8900922

SCHEMBL8900922

O=C1CCC(c2ccccc2)=C1O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CFTR P13569 1/20 0.46
GOPC Q9HD26 1/20 0.46
PTGS2 P35354 5/20 0.46
PTGS1 P23219 4/20 0.46
KMT2A Q03164 1/20 0.41
ALDH1A1 P00352 2/20 0.39
HTT P42858 2/20 0.39
P2RX7 Q99572 1/20 0.38
HDAC4 P56524 2/20 0.38
HDAC2 Q92769 2/20 0.38
HDAC8 Q9BY41 2/20 0.38
HDAC6 Q9UBN7 1/20 0.38
KDM4E B2RXH2 1/20 0.36
HPGD P15428 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
LMNA P02545 1/20 0.36
MAPT P10636 1/20 0.36
MMP3 P08254 1/20 0.36
BCL2L1 Q07817 1/20 0.36
FGF23 Q9GZV9 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL978197 0.77 PTGS2 (0.68) CFTRGOPCPTGS2PTGS1KMT2A
SCHEMBL5395859 0.76 CFTR (0.48) CFTRGOPCPTGS2PTGS1KMT2A
SCHEMBL5413521 0.74 CFTR (0.46) CFTRGOPCPTGS2PTGS1KMT2A
SCHEMBL31678688 0.74 PTGS2 (0.50) CFTRGOPCPTGS2PTGS1KMT2A
SCHEMBL28293315 0.74 CFTR (0.46) CFTRGOPCPTGS2PTGS1KMT2A
SCHEMBL7212942 0.72 ALDH1A1 (0.53) CFTRGOPCPTGS2PTGS1KMT2A
SCHEMBL6632882 0.72 PTGS2 (0.62) CFTRGOPCPTGS2PTGS1KMT2A
SCHEMBL6566571 0.72 CFTR (0.42) CFTRGOPCPTGS2PTGS1KMT2A
SCHEMBL10298881 0.68 PTGS2 (0.66) PTGS2PTGS1KMT2AALDH1A1HPGD
SCHEMBL7577906 0.68 PTGS2 (0.61) CFTRGOPCPTGS2PTGS1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5684205-A CHLORIDE CHANNEL BLOCKERS FOR CONTROLLING AIRWAY DISEASES, SECRETORY DIARRHEA AND ANTIINFLAMMATORY AGENTS BAYER AKTIENGESELLSCHAFT (DE) 1997-11-04 US disclosed
EP-0701988-A1 Substituted cyclopentane-di- and triones, their preparation and their use as chloride channel blockers BAYER AG (DE) 1996-03-20 EP disclosed