SCHEMBL8901168

SCHEMBL8901168

CN1CCN(c2ccccc2OCCCCC(=O)N2CCC(Cc3ccccc3)CC2)CC1

nearest known ligand 0.56

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
AVPR2 P30518 1/20 0.54
AVPR1A P37288 1/20 0.54
SLC6A2 P23975 1/20 0.53
SLC6A4 P31645 1/20 0.53
KDM4E B2RXH2 3/20 0.49
ALDH1A1 P00352 2/20 0.49
NPSR1 Q6W5P4 1/20 0.49
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
POLB P06746 1/20 0.48
HTR1A P08908 2/20 0.48
HTR7 P34969 2/20 0.48
DRD2 P14416 1/20 0.48
GAA P10253 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8901143 0.90 AVPR2 (0.52) AVPR2AVPR1AKDM4EALDH1A1MEN1
SCHEMBL8722874 0.85 AVPR2 (0.58) AVPR2AVPR1AKDM4EALDH1A1NPSR1
SCHEMBL8720267 0.85 AVPR2 (0.58) AVPR2AVPR1AKDM4EALDH1A1NPSR1
SCHEMBL8921897 0.84 AVPR2 (0.54) AVPR2AVPR1AKDM4EALDH1A1NPSR1
SCHEMBL8722383 0.83 HTR1A (0.58) AVPR2AVPR1AKDM4EALDH1A1HTR1A
SCHEMBL8907755 0.83 AVPR2 (0.53) AVPR2AVPR1AKDM4EALDH1A1NPSR1
SCHEMBL8722757 0.82 DRD2 (0.65) AVPR2AVPR1AKDM4EALDH1A1MEN1
SCHEMBL8901177 0.81 HTR1A (0.67) AVPR2AVPR1AKDM4EALDH1A1MEN1
SCHEMBL8724506 0.81 HTR1A (0.67) AVPR2AVPR1AKDM4EALDH1A1MEN1
SCHEMBL8902187 0.81 HTR1A (0.67) AVPR2AVPR1AKDM4EALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997014689-A1 ARYL-PIPERAZINE CYCLIC AMINE DERIVATIVES, PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME PIERRE FABRE MEDICAMENT (FR) 1997-04-24 WO disclosed