SCHEMBL8902889

SCHEMBL8902889

O=C(O)c1c(O)c(-c2ccc3ccccc3c2)cc2ccccc12

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.54
KDM4E B2RXH2 1/20 0.54
MEN1 O00255 1/20 0.54
ALDH1A1 P00352 1/20 0.54
GLA P06280 1/20 0.54
HPGD P15428 1/20 0.54
CYP2C19 P33261 1/20 0.54
KMT2A Q03164 1/20 0.54
HSD17B10 Q99714 1/20 0.54
GPR84 Q9NQS5 1/20 0.51
HDAC4 P56524 1/20 0.50
HDAC2 Q92769 1/20 0.50
HDAC8 Q9BY41 1/20 0.50
ACMSD Q8TDX5 2/20 0.49
ME2 P23368 1/20 0.47
ME1 P48163 1/20 0.47
ME3 Q16798 1/20 0.47
GSTP1 P09211 1/20 0.46
DHODH Q02127 5/20 0.46
MCL1 Q07820 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8440978 0.88 MEN1 (0.58) CYP1A2KDM4EMEN1ALDH1A1GLA
SCHEMBL338938 0.87 MEN1 (0.61) CYP1A2KDM4EMEN1ALDH1A1GLA
SCHEMBL10783912 0.83 CYP1A2 (0.55) CYP1A2KDM4EMEN1ALDH1A1GLA
SCHEMBL25439101 0.80 HDAC4 (0.54) CYP1A2KDM4EMEN1ALDH1A1HPGD
SCHEMBL18575575 0.79 GPR84 (0.57) CYP1A2KDM4EMEN1ALDH1A1HPGD
SCHEMBL30421930 0.76 MEN1 (0.54) CYP1A2KDM4EMEN1ALDH1A1GLA
SCHEMBL1661025 0.76 MEN1 (0.54) CYP1A2KDM4EMEN1ALDH1A1GLA
SCHEMBL29779946 0.75 CYP1A2 (0.68) CYP1A2KDM4EMEN1ALDH1A1GLA
SCHEMBL88986 0.75 CYP1A2 (0.68) CYP1A2KDM4EMEN1ALDH1A1GLA
SCHEMBL5553181 0.75 MEN1 (0.49) CYP1A2KDM4EMEN1ALDH1A1GLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997048672-A2 SUBSTITUTED TETRAHYDRONAPHTHALENE AND DIHYDRONAPHTHALENE DERIVATIVES HAVING RETINOID AND/OR RETINOID ANTAGONIST-LIKE BIOLOGICAL ACTIVITY ALLERGAN SALES, INC. (US) 1997-12-24 WO disclosed