SCHEMBL8903606

SCHEMBL8903606

CC(C)(C)OC(=O)CC(CN)c1ccc(Cl)c(Cl)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABBR2 O75899 4/20 0.42
GABBR1 Q9UBS5 4/20 0.42
LMNA P02545 3/20 0.42
CYP2C9 P11712 2/20 0.42
CYP3A4 P08684 1/20 0.42
ADORA3 P0DMS8 1/20 0.42
NFKB1 P19838 1/20 0.42
DRD3 P35462 1/20 0.42
BLM P54132 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C19 P33261 1/20 0.42
MEN1 O00255 1/20 0.42
THRB P10828 1/20 0.42
TSHR P16473 1/20 0.42
KMT2A Q03164 1/20 0.42
GAA P10253 1/20 0.40
ALDH1A1 P00352 1/20 0.39
HTT P42858 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8903093 0.85 GAA (0.46) GABBR2GABBR1LMNACYP2C9CYP3A4
SCHEMBL8770867 0.83 ALDH1A1 (0.42) LMNAALDH1A1HTTSMN1; SMN2SLC6A3
SCHEMBL21656114 0.83 GABBR2 (0.41) GABBR2GABBR1LMNACYP2C9CYP3A4
SCHEMBL21656591 0.80 GABBR2 (0.43) GABBR2GABBR1LMNACYP2C9CYP3A4
SCHEMBL8903798 0.79 GABBR2 (0.40) GABBR2GABBR1LMNACYP2C9CYP3A4
SCHEMBL5877648 0.79 GABBR2 (0.42) GABBR2GABBR1LMNACYP2C9CYP3A4
SCHEMBL5877614 0.79 GABBR2 (0.42) GABBR2GABBR1LMNACYP2C9CYP3A4
SCHEMBL5877532 0.79 GABBR2 (0.42) GABBR2GABBR1LMNACYP2C9CYP3A4
SCHEMBL21656318 0.78 GABBR2 (0.42) GABBR2GABBR1GAA
SCHEMBL27494782 0.78 GABBR2 (0.42) GABBR2GABBR1CYP2D6GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5686609-A Aromatic amine compounds, Their method of preparation and pharmaceutical compositions in which they are present SANOFI (FR) 1997-11-11 US disclosed
US-5618938-A Process for preparing stereo isomers of neurokinin receptor antagonists SANOFI (FR) 1997-04-08 US disclosed
US-5317020-A Neurokinin receiver antagonist as antiinflammatory agents SANOFI (FR) 1994-05-31 US disclosed