SCHEMBL8905241

SCHEMBL8905241

Cc1nc2ncn(C)c(=O)c2[nH]1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 2/20 0.40
CYP3A4 P08684 2/20 0.39
PMP22 Q01453 2/20 0.39
LMNA P02545 2/20 0.39
ALDH1A1 P00352 1/20 0.39
MAPT P10636 1/20 0.39
TSHR P16473 1/20 0.39
BLM P54132 1/20 0.39
SYK P43405 2/20 0.37
GDA Q9Y2T3 2/20 0.36
PDE2A O00408 1/20 0.36
PDE1A P54750 1/20 0.36
PDE1B Q01064 1/20 0.36
PDE1C Q14123 1/20 0.36
MAPK1 P28482 1/20 0.35
AKT2 P31751 1/20 0.35
ADORA3 P0DMS8 3/20 0.33
TAF1 P21675 1/20 0.33
BRPF1 P55201 1/20 0.33
CREBBP Q92793 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL763929 0.76 GDA (0.50) CYP3A4PMP22LMNAALDH1A1MAPT
SCHEMBL13217355 0.74 AURKA (0.43) CYP3A4ALDH1A1TSHRSYKADORA1
SCHEMBL2115743 0.72 ALDH1A1 (0.52) CYP3A4PMP22LMNAALDH1A1MAPT
SCHEMBL8272432 0.69 BRD9 (0.47) BRD4CYP3A4PMP22LMNAALDH1A1
SCHEMBL8392030 0.69 PDE2A (0.41) BRD4CYP3A4PMP22LMNABLM
SCHEMBL7191707 0.68 PDE2A (0.40) BRD4CYP3A4PMP22LMNAALDH1A1
SCHEMBL20203174 0.67 ADORA2A (0.48) CYP3A4PMP22LMNAALDH1A1MAPT
Caffeine SCHEMBL2327080 0.66 ADORA2A (0.68) CYP3A4PMP22BLMGDAPDE2A
SCHEMBL9910656 0.66 XDH (0.42) CYP3A4PMP22GDAMAPK1ADORA3
SCHEMBL8906319 0.65 ALDH1A1 (0.59) ALDH1A1GDA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5698685-A Morpholino-subunit combinatorial library and method ANTIVIRALS INC. (US) 1997-12-16 US disclosed
US-5506337-A Morpholino-subunit combinatorial library and method ANTIVIRALS INC. (US) 1996-04-09 US disclosed