SCHEMBL8906709

SCHEMBL8906709

CCCCc1nc2ccc(-c3nc4cc(OC)ccc4n3C)cc2n1-c1ccc(-c2ccccc2)c(C(=O)O)c1C

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARG P37231 5/20 0.42
CNR2 P34972 1/20 0.40
DHODH Q02127 1/20 0.40
EDNRA P25101 1/20 0.39
ACSS2 Q9NR19 1/20 0.39
LMNA P02545 1/20 0.38
KDM4E B2RXH2 1/20 0.38
ABCC3 O15438 1/20 0.38
ABCC4 O15439 1/20 0.38
USP2 O75604 1/20 0.38
ABCB11 O95342 1/20 0.38
ALDH1A1 P00352 1/20 0.38
CHRM2 P08172 1/20 0.38
CYP3A4 P08684 1/20 0.38
ADRA2A P08913 1/20 0.38
ADORA3 P0DMS8 1/20 0.38
CHRM1 P11229 1/20 0.38
CYP2C9 P11712 1/20 0.38
ACE P12821 1/20 0.38
ADRA2C P18825 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8906713 0.91 AGTR1 (0.45) PPARGKDM4EABCC3ABCC4USP2
SCHEMBL8905585 0.89 PPARG (0.43) PPARGEDNRAKDM4EABCC3ABCC4
SCHEMBL8905974 0.86 PPARG (0.45) PPARGDHODHKDM4EABCC3ABCC4
SCHEMBL8906712 0.86 PPARG (0.49) PPARGKDM4EABCC3ABCC4USP2
SCHEMBL8905700 0.85 PPARG (0.50) PPARGKDM4EABCC3ABCC4USP2
SCHEMBL8906533 0.84 PPARG (0.43) PPARGDHODHKDM4EABCC3ABCC4
SCHEMBL8905384 0.84 PPARG (0.46) PPARGDHODHKDM4EABCC3ABCC4
SCHEMBL8905690 0.84 PPARG (0.47) PPARGKDM4EABCC3ABCC4USP2
SCHEMBL8906316 0.83 PPARG (0.44) PPARGDHODHKDM4EABCC3ABCC4
SCHEMBL8906956 0.83 ALDH1A1 (0.44) PPARGDHODHLMNAKDM4EABCC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5684029-A HYPOTENSIVE AGENTS KARL THOMAE GMBH (DE) 1997-11-04 US disclosed