SCHEMBL8908135

SCHEMBL8908135

Fc1ccc(C2CCC3(CCCC(c4ccc5ccccc5c4)C3)C2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 1/20 0.43
RCOR1 Q9UKL0 1/20 0.43
CYP1A2 P05177 3/20 0.38
TRPA1 O75762 1/20 0.38
CYP2A6 P11509 1/20 0.38
SLC6A4 P31645 10/20 0.37
SLC6A2 P23975 9/20 0.37
SLC6A3 Q01959 9/20 0.37
EGFR P00533 2/20 0.37
ERBB2 P04626 2/20 0.37
DRD2 P14416 1/20 0.36
KDM4E B2RXH2 1/20 0.36
CYP2D6 P10635 3/20 0.36
KCNH2 Q12809 1/20 0.36
ESR1 P03372 1/20 0.35
ESR2 Q92731 1/20 0.35
HTR2A P28223 1/20 0.35
HTR2C P28335 1/20 0.35
LSS P48449 1/20 0.33
CYP1A1 P04798 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8908131 0.91 KDM1A (0.46) KDM1ARCOR1CYP1A2CYP2A6SLC6A4
SCHEMBL8907343 0.79 TACR1 (0.49) KDM1ARCOR1TRPA1DRD2HTR2A
SCHEMBL21559944 0.78 TRPA1 (0.41) KDM1ARCOR1TRPA1SLC6A3ESR1
SCHEMBL8907499 0.75 ESR2 (0.44) KDM1ARCOR1TRPA1DRD2ESR1
SCHEMBL8907505 0.75 ESR2 (0.44) KDM1ARCOR1TRPA1DRD2ESR1
SCHEMBL5400233 0.71 SLC6A4 (0.56) SLC6A4SLC6A2SLC6A3DRD2KDM4E
SCHEMBL4648603 0.71 SLC6A4 (0.56) SLC6A4SLC6A2SLC6A3DRD2KDM4E
SCHEMBL3673985 0.69 BACE1 (0.54) SLC6A4SLC6A2SLC6A3DRD2KDM4E
Naphthalene SCHEMBL9359039 0.69 BACE1 (0.54) SLC6A4SLC6A2SLC6A3DRD2KDM4E
SCHEMBL28228539 0.69 BACE1 (0.54) SLC6A4SLC6A2SLC6A3DRD2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0799231-A1 SPIROKETAL DERIVATIVES, COMPOSITIONS CONTAINING THEM AND THEIR USE AS THERAPEUTIC AGENTS MERCK SHARP & DOHME LTD. (GB) 1997-10-08 EP disclosed