SCHEMBL8908131

SCHEMBL8908131

Fc1ccc(C2CCC3(CC2)CCC(c2ccc4ccccc4c2)C3)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 1/20 0.46
RCOR1 Q9UKL0 1/20 0.46
SLC6A4 P31645 9/20 0.42
DRD2 P14416 1/20 0.42
CYP1A2 P05177 1/20 0.41
CYP2A6 P11509 1/20 0.41
SLC6A3 Q01959 8/20 0.40
SLC6A2 P23975 7/20 0.40
EGFR P00533 2/20 0.39
ERBB2 P04626 2/20 0.39
CYP2D6 P10635 1/20 0.38
KCNH2 Q12809 1/20 0.38
ESR2 Q92731 2/20 0.38
ESR1 P03372 1/20 0.38
HTR2A P28223 1/20 0.37
HTR2C P28335 1/20 0.37
KDM4E B2RXH2 1/20 0.36
GSK3B P49841 1/20 0.34
ADK P55263 1/20 0.34
MMP2 P08253 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8908135 0.91 KDM1A (0.43) KDM1ARCOR1SLC6A4DRD2CYP1A2
SCHEMBL8907505 0.85 ESR2 (0.44) KDM1ARCOR1DRD2ESR2ESR1
SCHEMBL8907499 0.85 ESR2 (0.44) KDM1ARCOR1DRD2ESR2ESR1
SCHEMBL8907338 0.77 HTR2C (0.52) KDM1ARCOR1DRD2HTR2AHTR2C
SCHEMBL5405317 0.74 SLC6A4 (0.59) KDM1ASLC6A4DRD2SLC6A3SLC6A2
SCHEMBL8907550 0.72 MEN1 (0.38) SLC6A4SLC6A3SLC6A2ESR2ESR1
SCHEMBL21559944 0.72 TRPA1 (0.41) KDM1ARCOR1SLC6A3ESR2ESR1
SCHEMBL5400233 0.70 SLC6A4 (0.56) SLC6A4DRD2SLC6A3SLC6A2CYP2D6
SCHEMBL4648603 0.70 SLC6A4 (0.56) SLC6A4DRD2SLC6A3SLC6A2CYP2D6
SCHEMBL8912656 0.69 TACR1 (0.46) KDM1ARCOR1SLC6A4DRD2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0799231-A1 SPIROKETAL DERIVATIVES, COMPOSITIONS CONTAINING THEM AND THEIR USE AS THERAPEUTIC AGENTS MERCK SHARP & DOHME LTD. (GB) 1997-10-08 EP disclosed