SCHEMBL8908139

SCHEMBL8908139

c1ccc2c(SCCCCCSc3ccnc4ccccc34)ccnc2c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.47
ADRA1D P25100 2/20 0.47
ADRA1A P35348 2/20 0.47
ADRA1B P35368 2/20 0.47
LOXL2 Q9Y4K0 1/20 0.46
NCF1 P14598 1/20 0.44
SLC22A12 Q96S37 1/20 0.42
FERMT2 Q96AC1 1/20 0.39
CYP2D6 P10635 2/20 0.39
CYP3A4 P08684 1/20 0.39
HIF1A Q16665 1/20 0.39
CYP1A2 P05177 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
KDM4E B2RXH2 2/20 0.38
MAPT P10636 1/20 0.38
ACP1 P24666 1/20 0.37
PRNP P04156 1/20 0.37
RXFP1 Q9HBX9 1/20 0.37
KCNH2 Q12809 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2333890 1.00 HTR1A (0.47) HTR1AADRA1DADRA1AADRA1BLOXL2
SCHEMBL12796611 0.84 LOXL2 (0.53) HTR1AADRA1DADRA1AADRA1BLOXL2
SCHEMBL14641227 0.80 HTR1A (0.46) HTR1AADRA1DADRA1AADRA1BLOXL2
SCHEMBL2816694 0.80 LOXL2 (0.47) HTR1AADRA1DADRA1AADRA1BLOXL2
SCHEMBL1147625 0.79 LOXL2 (0.43) HTR1AADRA1DADRA1AADRA1BLOXL2
SCHEMBL18548747 0.77 TLR8 (0.44) KDM4EMAPT
SCHEMBL13601938 0.77 HTR1A (0.43) HTR1AADRA1DADRA1AADRA1BLOXL2
SCHEMBL25404797 0.75 PIK3CA (0.45) SLC22A12CYP1A2
SCHEMBL25402921 0.75 ALK (0.44) CYP3A4KDM4EACP1PRNPRXFP1
SCHEMBL1147520 0.75 KDM4E (0.65) SLC22A12CYP1A2CYP2C9KDM4EPRNP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997048705-A1 POTASSIUM CHANNEL BLOCKERS UNIVERSITY COLLEGE LONDON (GB) 1997-12-24 WO disclosed