SCHEMBL8908353

SCHEMBL8908353

O=C1C=C(Nc2ccc(Cl)cc2)CC1

nearest known ligand 0.83

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MT-CO2 P00403 1/20 0.83
KMT2A Q03164 4/20 0.58
MAPT P10636 2/20 0.58
KDM4E B2RXH2 1/20 0.58
CYP1A2 P05177 1/20 0.58
CYP3A4 P08684 1/20 0.58
CYP2D6 P10635 1/20 0.58
CYP2C9 P11712 1/20 0.58
HPGD P15428 1/20 0.58
MAPK1 P28482 1/20 0.58
CYP2C19 P33261 1/20 0.58
NPSR1 Q6W5P4 1/20 0.58
POLB P06746 4/20 0.54
LMNA P02545 2/20 0.54
MEN1 O00255 3/20 0.47
ALDH1A1 P00352 2/20 0.42
IDO1 P14902 1/20 0.42
DHODH Q02127 1/20 0.41
ALOX15 P16050 1/20 0.40
HSD17B10 Q99714 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10811051 0.82 MT-CO2 (0.58) MT-CO2KMT2AMAPTKDM4ECYP1A2
SCHEMBL17481769 0.75 MT-CO2 (0.51) MT-CO2KMT2AMAPTKDM4ECYP1A2
SCHEMBL8906567 0.75 MAPK1 (0.66) MT-CO2KMT2AMAPTKDM4ECYP1A2
SCHEMBL486586 0.75 ALDH1A1 (0.72) MT-CO2KMT2AKDM4EPOLBMEN1
SCHEMBL16539324 0.74 MT-CO2 (0.50) MT-CO2KMT2AMAPTKDM4EPOLB
SCHEMBL16539777 0.73 POLB (0.69) MT-CO2KMT2AMAPTKDM4EHPGD
SCHEMBL16321423 0.72 MT-CO2 (0.48) MT-CO2KMT2AMAPTPOLBMEN1
SCHEMBL7522548 0.72 MT-CO2 (0.51) MT-CO2KMT2AMAPTKDM4ECYP1A2
SCHEMBL7520380 0.72 MT-CO2 (0.51) MT-CO2KMT2AMAPTKDM4ECYP1A2
SCHEMBL8906911 0.71 MT-CO2 (0.50) MT-CO2KMT2AMAPTKDM4ECYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5616615-A ANTICONVULSANTS HOWARD UNIVERSITY (US) 1997-04-01 US disclosed
US-5468775-A Anticonvulsants HOWARD UNIVERSITY (US) 1995-11-21 US disclosed
WO-1993017678-A1 ENAMINONE ESTERS HOWARD UNIVERSITY (US) 1993-09-16 WO disclosed