SCHEMBL8906911

SCHEMBL8906911

COC(=O)C1CCC(Nc2ccc(Cl)cc2)=CC1=O

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MT-CO2 P00403 1/20 0.50
KMT2A Q03164 3/20 0.40
MAPT P10636 2/20 0.40
ALDH1A1 P00352 1/20 0.40
KDM4E B2RXH2 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
HPGD P15428 1/20 0.40
MAPK1 P28482 1/20 0.40
CYP2C19 P33261 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
LMNA P02545 3/20 0.39
POLB P06746 3/20 0.39
IDO1 P14902 1/20 0.37
MEN1 O00255 2/20 0.36
AKR1C3 P42330 1/20 0.35
AKR1C2 P52895 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6545141 0.75 ALDH1A1 (0.52) MT-CO2KMT2AMAPTALDH1A1KDM4E
SCHEMBL29377973 0.75 ALDH1A1 (0.52) MT-CO2KMT2AMAPTALDH1A1KDM4E
SCHEMBL8908353 0.71 MT-CO2 (0.83) MT-CO2KMT2AMAPTALDH1A1KDM4E
SCHEMBL29958702 0.68 F7 (0.40) KMT2AMAPTALDH1A1KDM4EHPGD
SCHEMBL27033724 0.68 F7 (0.40) KMT2AMAPTALDH1A1KDM4EHPGD
SCHEMBL3393144 0.67 L3MBTL1 (0.47) KMT2AMAPTALDH1A1KDM4ECYP1A2
SCHEMBL13920758 0.66 PSEN1 (0.32) MAPTALDH1A1KDM4ECYP1A2CYP2C9
SCHEMBL23670494 0.65 P2RX7 (0.46) ALDH1A1AKR1C3
SCHEMBL5896818 0.65 GPBAR1 (0.48)
SCHEMBL29552779 0.65 P2RX7 (0.46) ALDH1A1AKR1C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5616615-A ANTICONVULSANTS HOWARD UNIVERSITY (US) 1997-04-01 US disclosed
US-5468775-A Anticonvulsants HOWARD UNIVERSITY (US) 1995-11-21 US disclosed
WO-1993017678-A1 ENAMINONE ESTERS HOWARD UNIVERSITY (US) 1993-09-16 WO disclosed