SCHEMBL8909616

SCHEMBL8909616

Oc1ccc(Cl)c2c1CCNCC2

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 7/20 0.50
HTR2A P28223 6/20 0.50
HTR2B P41595 6/20 0.50
PNMT P11086 4/20 0.42
ADRA2A P08913 1/20 0.40
ADRA2B P18089 1/20 0.40
ADRA2C P18825 1/20 0.40
ADCY6 O43306 1/20 0.40
ADCY3 O60266 1/20 0.40
ADCY9 O60503 1/20 0.40
ADCY5 O95622 1/20 0.40
ADCY8 P40145 1/20 0.40
ADCY7 P51828 1/20 0.40
ADCY2 Q08462 1/20 0.40
ADCY1 Q08828 1/20 0.40
ADCY4 Q8NFM4 1/20 0.40
NOTUM Q6P988 1/20 0.38
CYP3A4 P08684 1/20 0.38
MAPK1 P28482 1/20 0.38
HTR7 P34969 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16518065 0.88 PNMT (0.53) HTR2CHTR2AHTR2BPNMTADRA2A
Chlorindanol SCHEMBL29929703 0.80 CYP3A4 (0.42) HTR2CHTR2AHTR2BCYP3A4MAPK1
Chlorindanol SCHEMBL615288 0.80 CYP3A4 (0.42) HTR2CHTR2AHTR2BCYP3A4MAPK1
SCHEMBL10773279 0.80 BCL2L1 (0.45) CYP3A4MAPK1
SCHEMBL6188234 0.76 PNMT (0.63) HTR2CHTR2AHTR2BPNMTADRA2A
SCHEMBL20977986 0.75 HTR2C (0.50) HTR2CHTR2AHTR2BPNMTADRA2A
SCHEMBL15055797 0.75 HTR2C (0.47) HTR2CHTR2AHTR2BADCY6ADCY3
Hydrochloric Acid SCHEMBL17965631 0.74 PNMT (0.61) HTR2CHTR2AHTR2BPNMTADRA2A
SCHEMBL8909950 0.73 HTR2A (0.49) HTR2CHTR2AHTR2BPNMTADRA2A
SCHEMBL8910486 0.72 ADRA2A (0.55) ADRA2AADRA2BADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5639748-A HYPOTENSIVE AGENTS SMITHKLINE BEECHAM CORPORATION (US) 1997-06-17 US disclosed
EP-0630372-A1 HETEROALKOXY BENZAZEPINES SMITHKLINE BEECHAM CORPORATION (US) 1994-12-28 EP disclosed
EP-0603314-A4 CHEMICAL COMPOUNDS. SMITHKLINE BEECHAM CORP (US) 1994-08-24 EP disclosed
EP-0630372-A4 HETEROALKOXY BENZAZEPINES. SMITHKLINE BEECHAM CORP (US) 1994-07-05 EP disclosed
EP-0603314-A1 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1994-06-29 EP disclosed
WO-1993004686-A1 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1993-03-18 WO disclosed
WO-1993003015-A1 HETEROALKOXY BENZAZEPINES SMITHKLINE BEECHAM CORPORATION (US) 1993-02-18 WO disclosed