SCHEMBL8910112

SCHEMBL8910112

O=C(O)c1[nH]c2cc(Cl)ccc2c1Cl

nearest known ligand 0.65

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GPR17 Q13304 1/20 0.61
KDM4E B2RXH2 1/20 0.57
MEN1 O00255 1/20 0.57
LMNA P02545 1/20 0.57
CYP2C9 P11712 1/20 0.57
HPGD P15428 1/20 0.57
MAPK1 P28482 1/20 0.57
BLM P54132 1/20 0.57
KMT2A Q03164 1/20 0.57
GRIN2D O15399 1/20 0.55
GRIN3B O60391 1/20 0.55
GRIN1 Q05586 1/20 0.55
GRIN2A Q12879 1/20 0.55
GRIN2B Q13224 1/20 0.55
GRIN2C Q14957 1/20 0.55
GRIN3A Q8TCU5 1/20 0.55
MAP2 P11137 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6921821 0.86 MAP2 (0.65) GPR17KDM4EMEN1LMNAKMT2A
SCHEMBL1144990 0.84 GPR17 (0.60) GPR17KDM4EMEN1LMNACYP2C9
SCHEMBL9449344 0.84 GPR17 (0.60) GPR17KDM4EMEN1LMNACYP2C9
SCHEMBL8752546 0.83 GPR17 (0.58) GPR17KDM4EMEN1LMNACYP2C9
SCHEMBL27784165 0.83 GPR17 (0.47) GPR17KDM4EMEN1LMNAHPGD
SCHEMBL4333071 0.83 GPR17 (0.58) GPR17KDM4EMEN1LMNACYP2C9
SCHEMBL21341417 0.83 GPR17 (0.58) GPR17MEN1CYP2C9KMT2A
SCHEMBL31025926 0.80 GPR17 (0.72) GPR17
SCHEMBL31025899 0.80 ALOX15 (0.65) GPR17KDM4EMEN1LMNACYP2C9
SCHEMBL9187231 0.79 GPR17 (0.74) GPR17

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5688946-A DIPEPTIDES FOR HYPOTENSIVE AGENTS AND CARDIOVASCULAR DISORDERS HOFFMANN LA ROCHE INC. (US) 1997-11-18 US disclosed
EP-0416373-A2 Amino acid derivatives F. HOFFMANN-LA ROCHE AG (CH) 1991-03-13 EP disclosed