SCHEMBL8912908

SCHEMBL8912908

CCOC(=O)[C@@H](CN)c1ccccc1

nearest known ligand 0.60

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MMP8 P22894 1/20 0.53
GAA P10253 1/20 0.51
PIN1 Q13526 1/20 0.49
MEN1 O00255 1/20 0.47
NPC1 O15118 1/20 0.47
KMT2A Q03164 1/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
CYP1A2 P05177 1/20 0.47
CYP2D6 P10635 1/20 0.47
PKM P14618 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
KDM4E B2RXH2 2/20 0.46
TSHR P16473 1/20 0.45
GABBR2 O75899 1/20 0.44
GABBR1 Q9UBS5 1/20 0.44
CHRM1 P11229 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL512129 1.00 MMP8 (0.53) MMP8GAAPIN1MEN1NPC1
Hydrochloric Acid SCHEMBL3449917 0.98 PIN1 (0.51) MMP8GAAPIN1MEN1NPC1
SCHEMBL28470487 0.86 MMP8 (0.50) MMP8GAAPIN1MEN1NPC1
SCHEMBL5200954 0.86 LMNA (0.50) MEN1KMT2ASMN1; SMN2CYP1A2CYP2D6
Hydrazine SCHEMBL27358872 0.86 GAA (0.59) MMP8GAAMEN1KMT2AKDM4E
SCHEMBL23027214 0.85 GAA (0.62) MMP8GAAPIN1MEN1KMT2A
SCHEMBL260296 0.85 GAA (0.62) MMP8GAAPIN1MEN1KMT2A
SCHEMBL5972492 0.85 MMP8 (0.56) MMP8GAAPIN1MEN1NPC1
SCHEMBL805646 0.85 GAA (0.62) MMP8GAAPIN1MEN1KMT2A
SCHEMBL11641330 0.84 ESR1 (0.49) GAAKMT2ASMN1; SMN2CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0808303-A1 5-(4-SUBST.-PIPERIDINYL-1)-3-ARYL-PENTANOIC ACID DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONIST ZENECA LIMITED (GB) 1997-11-26 EP disclosed
WO-1996024582-A1 5-(4-SUBST.-PIPERIDINYL-1)-3-ARYL-PENTANOIC ACID DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONIST ZENECA LIMITED (GB) 1996-08-15 WO disclosed