SCHEMBL8912928

SCHEMBL8912928

CCc1c(C)[nH]c2cccc(O)c12

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 3/20 0.65
HTR2C P28335 2/20 0.65
HTT P42858 2/20 0.47
IMPDH2 P12268 1/20 0.46
IMPDH1 P20839 1/20 0.46
ALDH1A1 P00352 2/20 0.41
TSHR P16473 1/20 0.41
KDM4E B2RXH2 2/20 0.40
POLB P06746 1/20 0.40
SLC2A1 P11166 1/20 0.40
MAPT P10636 2/20 0.39
GAA P10253 1/20 0.39
CASP1 P29466 1/20 0.39
CASP7 P55210 1/20 0.39
CYP3A4 P08684 1/20 0.39
EP300 Q09472 1/20 0.38
CREBBP Q92793 1/20 0.38
BRD9 Q9H8M2 1/20 0.38
DAO P14920 1/20 0.38
DDO Q99489 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1920877 0.81 HTT (0.50) HTR2AHTR2CHTTALDH1A1TSHR
SCHEMBL2009406 0.80 KDM4E (0.60) HTR2AHTR2CIMPDH2IMPDH1ALDH1A1
SCHEMBL31060568 0.79 HTR2A (1.00) HTR2AHTR2CHTTIMPDH2IMPDH1
SCHEMBL18509955 0.78 HTR2A (0.63) HTR2AHTR2CALDH1A1KDM4EPOLB
SCHEMBL933915 0.77 HTR2A (0.54) HTR2AHTR2CIMPDH2IMPDH1TSHR
SCHEMBL11248441 0.77 HTR2A (0.55) HTR2AHTR2CHTTIMPDH2IMPDH1
SCHEMBL18029085 0.75 HTR2A (0.52) HTR2AHTR2CALDH1A1TSHRKDM4E
SCHEMBL14981556 0.72 FBP1 (0.46) HTR2AHTR2CHTTALDH1A1TSHR
Chloroform SCHEMBL11530972 0.71 HTR2A (0.49) HTR2AHTR2CIMPDH2IMPDH1ALDH1A1
SCHEMBL7747845 0.71 HTR2A (0.43) HTR2AHTR2CIMPDH2IMPDH1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0793656-A1 NOVEL BENZYL PYRIMIDINES F. HOFFMANN-LA ROCHE AG (CH) 1997-09-10 EP claimed
WO-1996016046-A2 NOVEL BENZYL PYRIMIDINES F. HOFFMANN-LA ROCHE AG (CH) 1996-05-30 WO claimed