SCHEMBL8913100

SCHEMBL8913100

CCOC(=O)CC(CC(=O)N(C)Cc1ccccc1OC)c1ccc(Cl)c(Cl)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
CRHBP P24387 1/20 0.46
CRHR2 Q13324 1/20 0.46
GAA P10253 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
NPC1 O15118 1/20 0.42
TACR1 P25103 2/20 0.40
BCHE P06276 5/20 0.39
ACHE P22303 5/20 0.39
TACR3 P29371 1/20 0.39
SLC6A4 P31645 4/20 0.39
SLC6A2 P23975 3/20 0.39
SLC6A3 Q01959 3/20 0.39
CHRM2 P08172 1/20 0.39
CHRM1 P11229 1/20 0.39
KCNH2 Q12809 2/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
HTR2A P28223 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6975177 0.89 MEN1 (0.51) MEN1KMT2ACRHBPCRHR2GAA
SCHEMBL6973685 0.86 MEN1 (0.47) MEN1KMT2ACRHBPCRHR2GAA
SCHEMBL6961996 0.85 MEN1 (0.47) MEN1KMT2ACRHBPCRHR2GAA
SCHEMBL7728008 0.79 SLC6A3 (0.49) SLC6A4SLC6A2SLC6A3
SCHEMBL7811404 0.76 TACR1 (0.49) MEN1KMT2ATDP1NPC1TACR1
SCHEMBL7728006 0.75 FFAR1 (0.50) SLC6A4SLC6A2SLC6A3
SCHEMBL7815283 0.74 KDM4E (0.45)
SCHEMBL7811403 0.73 TACR1 (0.46) MEN1KMT2ATDP1NPC1TACR1
SCHEMBL7871897 0.73 TACR2 (0.65) TACR1TACR3
SCHEMBL7873231 0.73 TACR2 (0.65) TACR1TACR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0808303-A1 5-(4-SUBST.-PIPERIDINYL-1)-3-ARYL-PENTANOIC ACID DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONIST ZENECA LIMITED (GB) 1997-11-26 EP disclosed
WO-1996024582-A1 5-(4-SUBST.-PIPERIDINYL-1)-3-ARYL-PENTANOIC ACID DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONIST ZENECA LIMITED (GB) 1996-08-15 WO disclosed