SCHEMBL8913460

SCHEMBL8913460

OC1=CC2(CCN(CCc3ccccn3)CC2)Sc2sccc21

nearest known ligand 0.47

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ADRA1D P25100 3/20 0.43
ADRA1A P35348 2/20 0.43
ADRA1B P35368 1/20 0.43
OPRM1 P35372 2/20 0.39
SIGMAR1 Q99720 2/20 0.39
THRB P10828 2/20 0.39
KCNH2 Q12809 1/20 0.38
TP53 P04637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8914168 0.81 ADRA1D (0.44) ADRA1DADRA1AADRA1BOPRM1SIGMAR1
SCHEMBL8914759 0.78 ADRA1D (0.56) ADRA1DADRA1AADRA1BOPRM1SIGMAR1
Hydrochloric Acid SCHEMBL8912532 0.77 ADRA1D (0.55) ADRA1DADRA1AADRA1BOPRM1SIGMAR1
SCHEMBL16026529 0.69 THRB (0.61) ADRA1DADRA1AADRA1BTHRBTP53
SCHEMBL29922137 0.69 THRB (0.61) ADRA1DADRA1AADRA1BTHRBTP53
Hydrochloric Acid SCHEMBL8912509 0.69 ADRA1D (0.49) ADRA1DADRA1AADRA1BOPRM1SIGMAR1
SCHEMBL8912590 0.67 ADRA1D (0.53) ADRA1DADRA1AADRA1BOPRM1SIGMAR1
SCHEMBL12359541 0.67 THRB (0.56) ADRA1DADRA1AADRA1BOPRM1SIGMAR1
SCHEMBL868571 0.67 HRH3 (0.56) SIGMAR1THRBTP53
SCHEMBL9592086 0.66 HTR2C (0.45) ADRA1DADRA1AADRA1BTHRBTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5633247-A ANTIARRTHYMIA AGENT MERCK & CO., INC. (US) 1997-05-27 US disclosed
US-5206240-A Antiarrhythmia agents MERCK & CO., INC. (US) 1993-04-27 US disclosed
EP-0431943-A2 Nitrogen-containing spirocycles MERCK & CO. INC. (US) 1991-06-12 EP disclosed