SCHEMBL8914759

SCHEMBL8914759

O=C1CC2(CCN(CCc3ccccn3)CC2)Sc2sccc21

nearest known ligand 0.56

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ADRA1D P25100 3/20 0.56
ADRA1A P35348 2/20 0.56
ADRA1B P35368 1/20 0.56
OPRM1 P35372 2/20 0.44
SIGMAR1 Q99720 2/20 0.44
KCNH2 Q12809 1/20 0.43
HSD17B10 Q99714 1/20 0.41
THRB P10828 2/20 0.40
TP53 P04637 1/20 0.39
CYP2D6 P10635 1/20 0.37
CYP2C19 P33261 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8912532 0.99 ADRA1D (0.55) ADRA1DADRA1AADRA1BOPRM1SIGMAR1
Hydrochloric Acid SCHEMBL8913902 0.82 ADRA1D (0.60) ADRA1DADRA1AADRA1BOPRM1SIGMAR1
SCHEMBL8913652 0.80 ADRA1D (0.51) ADRA1DADRA1AADRA1BOPRM1SIGMAR1
SCHEMBL8912590 0.78 ADRA1D (0.53) ADRA1DADRA1AADRA1BOPRM1SIGMAR1
SCHEMBL8913460 0.78 ADRA1D (0.43) ADRA1DADRA1AADRA1BOPRM1SIGMAR1
Hydrochloric Acid SCHEMBL9854583 0.77 SIGMAR1 (0.38) OPRM1SIGMAR1KCNH2
SCHEMBL8914168 0.75 ADRA1D (0.44) ADRA1DADRA1AADRA1BOPRM1SIGMAR1
Hydrochloric Acid SCHEMBL8563648 0.71 ADRA1D (0.98) ADRA1DADRA1AADRA1BOPRM1SIGMAR1
SCHEMBL9592086 0.71 HTR2C (0.45) ADRA1DADRA1AADRA1BHSD17B10THRB
SCHEMBL16026529 0.70 THRB (0.61) ADRA1DADRA1AADRA1BHSD17B10THRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5633247-A ANTIARRTHYMIA AGENT MERCK & CO., INC. (US) 1997-05-27 US disclosed
US-5206240-A Antiarrhythmia agents MERCK & CO., INC. (US) 1993-04-27 US disclosed