SCHEMBL8913489

SCHEMBL8913489

CS(=O)(=O)c1ccc2c(c1)CCC1(CCN(CCCCCCO)CC1)O2

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 4/20 0.53
CYP2C9 P11712 2/20 0.53
CYP2D6 P10635 1/20 0.53
EPHX1 P07099 2/20 0.49
HTR2A P28223 5/20 0.48
DRD2 P14416 4/20 0.48
HTR2C P28335 3/20 0.48
KCNH2 Q12809 2/20 0.43
HRH3 Q9Y5N1 6/20 0.42
GPR119 Q8TDV5 2/20 0.40
HDAC3 O15379 1/20 0.38
HDAC4 P56524 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC7 Q8WUI4 1/20 0.38
HDAC2 Q92769 1/20 0.38
HDAC10 Q969S8 1/20 0.38
HDAC11 Q96DB2 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
HDAC9 Q9UKV0 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8566857 0.75 ADRA1D (0.47) HTR2ADRD2HTR2CKCNH2
SCHEMBL8563145 0.73 EPHX2 (0.51) EPHX2EPHX1HTR2AKCNH2
SCHEMBL12695212 0.72 EPHX2 (0.78) EPHX2CYP2C9CYP2D6EPHX1GPR119
Hydrochloric Acid SCHEMBL8912554 0.72 EPHX2 (0.52) EPHX2CYP2C9CYP2D6EPHX1HTR2A
SCHEMBL8565545 0.70 ADRA1D (0.66) KCNH2
SCHEMBL8564077 0.70 ADRA1D (0.66) KCNH2
SCHEMBL8010281 0.70 DRD2 (0.74) EPHX2EPHX1HTR2ADRD2HTR2C
SCHEMBL12695002 0.69 EPHX2 (1.00) EPHX2CYP2C9CYP2D6EPHX1GPR119
SCHEMBL19838801 0.68 HTR2A (0.71) EPHX2EPHX1HTR2ADRD2HTR2C
SCHEMBL8576957 0.66 DRD2 (0.67) HTR2ADRD2HTR2CKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5633247-A ANTIARRTHYMIA AGENT MERCK & CO., INC. (US) 1997-05-27 US disclosed
US-5206240-A Antiarrhythmia agents MERCK & CO., INC. (US) 1993-04-27 US disclosed