SCHEMBL8914175

SCHEMBL8914175

c1ccc(CN2CCCC3(Cc4ccccc4O3)C2)cc1

nearest known ligand 0.60

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 8/20 0.60
HDAC3 O15379 1/20 0.49
HDAC4 P56524 1/20 0.49
HDAC1 Q13547 1/20 0.49
HDAC7 Q8WUI4 1/20 0.49
HDAC2 Q92769 1/20 0.49
HDAC10 Q969S8 1/20 0.49
HDAC11 Q96DB2 1/20 0.49
HDAC8 Q9BY41 1/20 0.49
HDAC6 Q9UBN7 1/20 0.49
HDAC9 Q9UKV0 1/20 0.49
HDAC5 Q9UQL6 1/20 0.49
DRD2 P14416 3/20 0.48
HTR2A P28223 1/20 0.48
CYP2D6 P10635 4/20 0.48
CYP3A4 P08684 1/20 0.43
TSHR P16473 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11184048 0.99 SIGMAR1 (0.59) SIGMAR1HDAC3HDAC4HDAC1HDAC7
SCHEMBL11257702 0.92 SIGMAR1 (0.71) SIGMAR1HDAC3HDAC4HDAC1HDAC7
SCHEMBL863908 0.90 SIGMAR1 (0.71) SIGMAR1HDAC3HDAC4HDAC1HDAC7
SCHEMBL864155 0.83 SIGMAR1 (0.79) SIGMAR1HDAC3HDAC4HDAC1HDAC7
Hydrochloric Acid SCHEMBL11193368 0.82 SIGMAR1 (0.77) SIGMAR1HDAC3HDAC4HDAC1HDAC7
SCHEMBL11246888 0.79 DRD2 (0.72) SIGMAR1HDAC3HDAC4HDAC1HDAC7
SCHEMBL2344239 0.79 SIGMAR1 (0.56) SIGMAR1DRD2CYP2D6CYP3A4TSHR
SCHEMBL4211897 0.79 DRD2 (0.69) SIGMAR1HDAC3HDAC4HDAC1HDAC7
Hydrochloric Acid SCHEMBL10502428 0.78 SIGMAR1 (0.40) SIGMAR1HDAC3HDAC4HDAC1HDAC7
SCHEMBL6263041 0.76 SIGMAR1 (0.54) SIGMAR1DRD2CYP2D6CYP3A4TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5633247-A ANTIARRTHYMIA AGENT MERCK & CO., INC. (US) 1997-05-27 US disclosed
US-5206240-A Antiarrhythmia agents MERCK & CO., INC. (US) 1993-04-27 US disclosed
EP-0431943-A2 Nitrogen-containing spirocycles MERCK & CO. INC. (US) 1991-06-12 EP disclosed