SCHEMBL8914198

SCHEMBL8914198

Cc1cc(CON2C(=O)c3ccccc3C2=O)no1

nearest known ligand 0.63

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.63
RECQL P46063 2/20 0.63
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
L3MBTL1 Q9Y468 1/20 0.44
GAA P10253 1/20 0.44
ALDH1A1 P00352 4/20 0.43
GABRA5 P31644 2/20 0.43
GABRA1 P14867 1/20 0.43
HTT P42858 1/20 0.43
ATM Q13315 1/20 0.41
GRIN2B Q13224 3/20 0.40
GRIN1 Q05586 2/20 0.40
CYP1A2 P05177 1/20 0.39
CYP2C9 P11712 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8913973 0.77 MEN1 (0.54) MAPTRECQLMEN1KMT2AGAA
SCHEMBL1716167 0.76 MAPT (0.42) MAPTRECQLMEN1KMT2AGAA
SCHEMBL13140635 0.74 MEN1 (0.46) MAPTRECQLMEN1KMT2AGAA
SCHEMBL8914384 0.74 TAS2R8 (0.51) MAPTMEN1KMT2AL3MBTL1GAA
SCHEMBL6921729 0.74 MEN1 (0.48) MAPTRECQLMEN1KMT2AGAA
SCHEMBL15071827 0.72 MEN1 (0.47) MAPTRECQLMEN1KMT2AGAA
SCHEMBL6610647 0.71 MEN1 (0.44) MAPTRECQLMEN1KMT2AGAA
SCHEMBL2219482 0.71 ALDH1A1 (0.58) MAPTRECQLMEN1KMT2AGAA
SCHEMBL31119039 0.71 MEN1 (0.59) MAPTRECQLMEN1KMT2AGAA
SCHEMBL10815849 0.71 MEN1 (0.48) MAPTRECQLMEN1KMT2AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5604256-A (7-(5-(1,3-DIOXANE-5YL)METHOXYIMINO-2-METHYL-8-(2-METHYLBUTYR -OXY)3-OXO-1,2,3,5,6,7,8,8A-OCTAHYDRO-1-NAPHTHYL)-3-HYDROXY-5 -OXOHEPTANOIC ACID AND SALTS SANKYO COMPANY, LIMITED (JP) 1997-02-18 US disclosed
EP-0570245-B1 Octahydronaphthalene oxime derivatives for cholesterol biosynthesis inhibition, their preparation and use SANKYO CO (JP) 1996-10-30 EP disclosed
EP-0570245-A2 Octahydronaphthalene oxime derivatives for cholesterol biosynthesis inhibition, their preparation and use SANKYO COMPANY LIMITED (JP) 1993-11-18 EP disclosed